SCHEMBL6863147

SCHEMBL6863147

Nc1cc(C(=O)NC2CCc3ccccc32)cc2nc(-c3ccoc3)nn12

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CHRM4 P08173 4/20 0.46
PDE4A P27815 1/20 0.42
PDE4B Q07343 1/20 0.42
PDE4C Q08493 1/20 0.42
PDE4D Q08499 1/20 0.42
HPGDS O60760 1/20 0.41
HTT P42858 1/20 0.41
KDM4E B2RXH2 3/20 0.41
ADA P00813 1/20 0.40
TAS1R3 Q7RTX0 2/20 0.40
TAS1R1 Q7RTX1 2/20 0.40
CNR1 P21554 1/20 0.40
ALDH1A1 P00352 3/20 0.40
ROCK2 O75116 1/20 0.40
MEN1 O00255 1/20 0.40
HPGD P15428 1/20 0.40
KMT2A Q03164 1/20 0.40
RECQL P46063 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6870587 0.89 CHRM4 (0.49) CHRM4PDE4APDE4BPDE4CPDE4D
SCHEMBL6872383 0.82 ADORA2A (0.56) CHRM4PDE4APDE4BPDE4CPDE4D
SCHEMBL6863240 0.81 CHRM4 (0.55) CHRM4PDE4APDE4BPDE4CPDE4D
SCHEMBL6869838 0.81 ADORA2A (0.43) HTTKDM4EALDH1A1MEN1HPGD
SCHEMBL6873668 0.80 CHRM4 (0.47) CHRM4PDE4APDE4BPDE4CPDE4D
SCHEMBL6868029 0.79 CHRM4 (0.52) CHRM4PDE4APDE4BPDE4CPDE4D
SCHEMBL6869842 0.77 PLAU (0.48) HTTKDM4EALDH1A1MEN1HPGD
SCHEMBL6863099 0.74 ADORA2A (0.45)
SCHEMBL6871806 0.73 ADORA2A (0.42)
SCHEMBL6870707 0.72 KMT2A (0.43) ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347974-B1 AMINOTRIAZOLOPYRIDIINE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS HOFFMANN LA ROCHE (CH) 2004-11-03 EP disclosed