SCHEMBL6869036

SCHEMBL6869036

Nc1cc(C(=O)NCc2ccc(F)cc2)cc2nc(-c3ccccn3)nn12

nearest known ligand 0.56

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 1/20 0.56
GLA P06280 1/20 0.52
KLKB1 P03952 11/20 0.51
F2 P00734 6/20 0.51
F10 P00742 3/20 0.51
KLK1 P06870 1/20 0.51
HPGDS O60760 2/20 0.47
F12 P00748 2/20 0.47
EGLN1 Q9GZT9 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6867628 0.92 ADORA2A (0.60) ADORA2AKLKB1F2F10KLK1
SCHEMBL6871169 0.88 ADORA2A (0.54) ADORA2AKLKB1F2KLK1HPGDS
SCHEMBL6872074 0.83 ADORA2A (0.56) ADORA2AF2HPGDSF12
SCHEMBL6870348 0.83 ADORA2A (0.56) ADORA2AF12
SCHEMBL6871731 0.83 ADORA2A (0.64) ADORA2AKLKB1F2F10KLK1
SCHEMBL7114944 0.82 ADORA2A (0.54) ADORA2A
SCHEMBL6873737 0.82 L3MBTL1 (0.43) ADORA2AL3MBTL1
SCHEMBL6870133 0.81 ADORA2A (0.59) ADORA2AKLKB1F2F12
SCHEMBL6869989 0.80 ADORA2A (0.58) ADORA2AKLKB1F2F12
SCHEMBL6871283 0.79 PTGER2 (0.44) ADORA2AKLKB1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347974-B1 AMINOTRIAZOLOPYRIDIINE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS HOFFMANN LA ROCHE (CH) 2004-11-03 EP disclosed