SCHEMBL6869989

SCHEMBL6869989

CCCCNC(=O)c1cc(N)n2nc(-c3ccccn3)nc2c1

nearest known ligand 0.58

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 3/20 0.58
RXFP1 Q9HBX9 1/20 0.48
F12 P00748 4/20 0.46
SMN1; SMN2 Q16637 3/20 0.45
KDR P35968 1/20 0.42
CAMK2D Q13557 1/20 0.42
NAAA Q02083 1/20 0.42
F2 P00734 3/20 0.41
EGLN2 Q96KS0 1/20 0.41
HTT P42858 1/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
ATM Q13315 1/20 0.40
PLG P00747 1/20 0.39
PLAU P00749 1/20 0.39
KIT P10721 1/20 0.39
DDR1 Q08345 1/20 0.39
KLKB1 P03952 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6872486 0.96 ADORA2A (0.56) ADORA2ARXFP1F12SMN1; SMN2NAAA
SCHEMBL6866973 0.85 BACE1 (0.48) SMN1; SMN2CAMK2DNAAAEGLN2HTT
SCHEMBL6870133 0.85 ADORA2A (0.59) ADORA2AF12F2PLGPLAU
SCHEMBL6867628 0.84 ADORA2A (0.60) ADORA2AF12F2PLAUKLKB1
SCHEMBL6872186 0.83 SMN1; SMN2 (0.43) ADORA2ARXFP1SMN1; SMN2KDRNAAA
SCHEMBL6871382 0.82 ADORA2A (0.59) ADORA2AF12NPC1RAB9AKIT
SCHEMBL6867215 0.81 PLAU (0.47) SMN1; SMN2CAMK2DF2PLAU
SCHEMBL6870656 0.80 ADORA2A (0.59) ADORA2AF12F2ATM
SCHEMBL6869823 0.80 ADORA2A (0.56) ADORA2AF12F2PLGPLAU
SCHEMBL6872074 0.80 ADORA2A (0.56) ADORA2AF12F2PLAU

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347974-B1 AMINOTRIAZOLOPYRIDIINE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS HOFFMANN LA ROCHE (CH) 2004-11-03 EP disclosed