SCHEMBL6869174

SCHEMBL6869174

COc1cc(CNCC2CCC(Nc3nccc(N(C)C)n3)CC2)cc(OC)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 2/20 0.45
KCNH2 Q12809 1/20 0.45
AURKB Q96GD4 1/20 0.45
MCHR1 Q99705 7/20 0.40
ACHE P22303 3/20 0.40
BACE1 P56817 2/20 0.40
FGFR1 P11362 1/20 0.38
KDR P35968 1/20 0.38
EPHB4 P54760 1/20 0.38
ADRA2A P08913 3/20 0.38
NPY5R Q15761 1/20 0.38
PRKCQ Q04759 1/20 0.37
TSHR P16473 2/20 0.37
ALDH1A1 P00352 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
DRD2 P14416 1/20 0.37
DRD3 P35462 1/20 0.37
MAPK6 Q16659 1/20 0.36
ADRA1A P35348 1/20 0.36
HRH1 P35367 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6869172 1.00 CNR1 (0.45) CNR1KCNH2AURKBMCHR1ACHE
SCHEMBL6875802 0.91 ACHE (0.48) CNR1KCNH2AURKBMCHR1ACHE
SCHEMBL6875798 0.91 ACHE (0.48) CNR1KCNH2AURKBMCHR1ACHE
SCHEMBL6873488 0.88 ACHE (0.51) CNR1KCNH2AURKBMCHR1ACHE
SCHEMBL6868661 0.88 CNR1 (0.41) CNR1KCNH2AURKBMCHR1ACHE
SCHEMBL6875018 0.88 ACHE (0.43) CNR1KCNH2AURKBMCHR1ACHE
SCHEMBL6873495 0.88 ACHE (0.51) CNR1KCNH2AURKBMCHR1ACHE
SCHEMBL6868672 0.88 CNR1 (0.41) CNR1KCNH2AURKBMCHR1ACHE
SCHEMBL6875044 0.88 ACHE (0.43) CNR1KCNH2AURKBMCHR1ACHE
SCHEMBL6873081 0.88 TSHR (0.51) CNR1KCNH2AURKBMCHR1ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1464335-A2 Quinoline, tetrahydroquinoline and pyrimidine derivatives as mch antagonist Taisho Pharmaceutical Co. Ltd. (JP) 2004-10-06 EP disclosed