SCHEMBL6868672

SCHEMBL6868672

COc1cc(OC)c(CNCC2CCC(Nc3nccc(N(C)C)n3)CC2)c(OC)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 1/20 0.41
KCNH2 Q12809 1/20 0.41
AURKB Q96GD4 1/20 0.41
MCHR1 Q99705 8/20 0.39
CD274 Q9NZQ7 1/20 0.39
ADRA2A P08913 3/20 0.39
NPY5R Q15761 1/20 0.39
ACHE P22303 3/20 0.37
BACE1 P56817 2/20 0.37
DRD2 P14416 2/20 0.37
DRD3 P35462 2/20 0.37
MAPK8 P45983 1/20 0.35
MAPK9 P45984 1/20 0.35
MAPK10 P53779 1/20 0.35
MAPK6 Q16659 1/20 0.35
ADRA1A P35348 1/20 0.35
HRH1 P35367 1/20 0.35
HTR2B P41595 1/20 0.35
FGFR1 P11362 1/20 0.35
KDR P35968 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6868661 1.00 CNR1 (0.41) CNR1KCNH2AURKBMCHR1CD274
SCHEMBL6877408 0.90 MAPK8 (0.42) KCNH2AURKBMCHR1CD274ADRA2A
SCHEMBL6457586 0.90 MAPK8 (0.42) KCNH2AURKBMCHR1CD274ADRA2A
SCHEMBL6874596 0.90 APLNR (0.44) CNR1KCNH2AURKBMCHR1ADRA2A
SCHEMBL6459873 0.90 APLNR (0.44) CNR1KCNH2AURKBMCHR1ADRA2A
SCHEMBL6869172 0.88 CNR1 (0.45) CNR1KCNH2AURKBMCHR1ADRA2A
SCHEMBL6869174 0.88 CNR1 (0.45) CNR1KCNH2AURKBMCHR1ADRA2A
SCHEMBL6875669 0.87 MCHR1 (0.41) CNR1KCNH2AURKBMCHR1ADRA2A
SCHEMBL6875677 0.87 MCHR1 (0.41) CNR1KCNH2AURKBMCHR1ADRA2A
SCHEMBL6873584 0.85 MCHR1 (0.42) CNR1KCNH2AURKBMCHR1ADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1464335-A2 Quinoline, tetrahydroquinoline and pyrimidine derivatives as mch antagonist Taisho Pharmaceutical Co. Ltd. (JP) 2004-10-06 EP disclosed