SCHEMBL6870096

SCHEMBL6870096

Cc1ccc(-c2nc3cc(C(=O)NCc4ccccc4)cc(N)n3n2)o1

nearest known ligand 0.60

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 16/20 0.60
PTPN22 Q9Y2R2 1/20 0.47
KDM4E B2RXH2 1/20 0.46
ALDH1A1 P00352 1/20 0.46
HPGD P15428 1/20 0.46
HSD17B10 Q99714 1/20 0.46
LMNA P02545 1/20 0.45
MAPK1 P28482 1/20 0.45
PLAU P00749 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6871992 0.90 ADORA2A (0.58) ADORA2AALDH1A1HPGDLMNA
SCHEMBL6871192 0.90 ADORA2A (0.58) ADORA2ALMNA
SCHEMBL6873589 0.89 ADORA2A (0.56) ADORA2AKDM4EALDH1A1HPGDLMNA
SCHEMBL6871493 0.88 ADORA2A (0.66) ADORA2AHPGDPLAU
SCHEMBL6871404 0.88 ADORA2A (0.51) ADORA2AKDM4EALDH1A1HPGDHSD17B10
SCHEMBL6873996 0.85 ADORA2A (0.55) ADORA2AKDM4EALDH1A1HPGDLMNA
SCHEMBL6868316 0.85 ADORA2A (0.55) ADORA2AKDM4EALDH1A1HPGDHSD17B10
SCHEMBL6867257 0.85 ADORA2A (0.55) ADORA2AALDH1A1HSD17B10
SCHEMBL6867554 0.85 ADORA2A (0.63) ADORA2AALDH1A1
SCHEMBL6873157 0.83 HPGDS (0.51) ADORA2AKDM4EALDH1A1HPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347974-B1 AMINOTRIAZOLOPYRIDIINE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS HOFFMANN LA ROCHE (CH) 2004-11-03 EP disclosed