SCHEMBL6867554

SCHEMBL6867554

Cc1ccc(-c2nc3cc(C(=O)Nc4ccccc4)cc(N)n3n2)o1

nearest known ligand 0.63

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 19/20 0.63
MEN1 O00255 1/20 0.43
ALDH1A1 P00352 1/20 0.43
POLB P06746 1/20 0.43
MAPT P10636 1/20 0.43
PKM P14618 1/20 0.43
KMT2A Q03164 1/20 0.43
HDAC1 Q13547 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6873045 0.88 ADORA2A (0.62) ADORA2AMEN1MAPTKMT2A
SCHEMBL6870096 0.85 ADORA2A (0.60) ADORA2AALDH1A1
SCHEMBL6863170 0.84 ADORA2A (0.73) ADORA2A
SCHEMBL6873028 0.82 ADORA2A (0.73) ADORA2A
SCHEMBL6868100 0.82 ADORA2A (0.44) ADORA2AMEN1ALDH1A1POLBMAPT
SCHEMBL6870475 0.81 ADORA2A (0.69) ADORA2AALDH1A1POLBPKM
SCHEMBL6870449 0.80 RAB9A (0.45) ADORA2AMEN1ALDH1A1MAPTKMT2A
SCHEMBL6870649 0.80 ADORA2A (0.61) ADORA2A
SCHEMBL6867550 0.79 ADORA2A (0.67) ADORA2A
SCHEMBL6873996 0.78 ADORA2A (0.55) ADORA2AALDH1A1POLBMAPTHDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347974-B1 AMINOTRIAZOLOPYRIDIINE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS HOFFMANN LA ROCHE (CH) 2004-11-03 EP disclosed