SCHEMBL687038

SCHEMBL687038

CCOc1ccc([C@H](CC(=O)O)NC(=O)Nc2c(O)c(C)nn(Cc3ccccc3Cl)c2=O)cc1OCC

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 5/20 0.43
KMT2A Q03164 4/20 0.40
CYP26A1 O43174 1/20 0.39
USP2 O75604 3/20 0.39
THRB P10828 1/20 0.39
NPSR1 Q6W5P4 8/20 0.39
POLB P06746 2/20 0.38
LMNA P02545 4/20 0.38
MEN1 O00255 3/20 0.38
GAA P10253 3/20 0.37
MAPK1 P28482 1/20 0.37
ALDH1A1 P00352 2/20 0.37
PDE4A P27815 1/20 0.37
PDE4B Q07343 1/20 0.37
PDE4C Q08493 1/20 0.37
PDE4D Q08499 1/20 0.37
KDM4E B2RXH2 1/20 0.37
HPGD P15428 1/20 0.37
HSD17B10 Q99714 1/20 0.37
MAPT P10636 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL687999 0.90 SLC16A3 (0.42) SMN1; SMN2KMT2ACYP26A1USP2THRB
SCHEMBL686977 0.89 SLC16A3 (0.42) SMN1; SMN2KMT2ACYP26A1USP2THRB
SCHEMBL688267 0.87 CTSA (0.43) SMN1; SMN2KMT2ACYP26A1NPSR1LMNA
SCHEMBL688254 0.86 SMN1; SMN2 (0.44) SMN1; SMN2KMT2ANPSR1POLBLMNA
SCHEMBL687242 0.86 SMN1; SMN2 (0.44) SMN1; SMN2KMT2ANPSR1POLBLMNA
SCHEMBL687862 0.84 SMN1; SMN2 (0.43) SMN1; SMN2KMT2ANPSR1POLBLMNA
SCHEMBL687629 0.83 SMN1; SMN2 (0.45) SMN1; SMN2KMT2ANPSR1POLBLMNA
SCHEMBL688067 0.83 SLC22A12 (0.39) SMN1; SMN2KMT2ACYP26A1NPSR1LMNA
SCHEMBL686627 0.83 SMN1; SMN2 (0.42) SMN1; SMN2KMT2ANPSR1POLBLMNA
SCHEMBL687875 0.83 CTSA (0.40) SMN1; SMN2CYP26A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1203766-B1 Carboxylic acid derivatives that inhibit the binding of integrins to their receptors ENCYSIVE PHARMACEUTICALS INC (US) 2012-02-29 EP disclosed
EP-1203766-A2 Carboxylic acid derivatives that inhibit the binding of integrins to their receptors TEXAS BIOTECHNOLOGY CORPORATION (US) 2002-05-08 EP disclosed