SCHEMBL6863096

SCHEMBL6863096

Nc1cc(C(=O)NCc2ccccc2Cl)cc2nc(-c3ccoc3)nn12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 5/20 0.43
ADORA2A P29274 2/20 0.43
ADORA1 P30542 2/20 0.43
TP53 P04637 3/20 0.42
ALDH1A1 P00352 3/20 0.42
KMT2A Q03164 2/20 0.42
ADORA3 P0DMS8 1/20 0.42
ADORA2B P29275 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
GAA P10253 1/20 0.42
TSHR P16473 1/20 0.42
CYP2C19 P33261 1/20 0.42
SCN2A Q99250 1/20 0.42
SCN10A Q9Y5Y9 1/20 0.42
LMNA P02545 4/20 0.41
HPGD P15428 2/20 0.41
HTT P42858 1/20 0.41
HSD17B10 Q99714 1/20 0.41
MAPT P10636 3/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6870707 0.89 KMT2A (0.43) ADORA2AALDH1A1KMT2ALMNAMAPT
SCHEMBL6863739 0.88 SMN1; SMN2 (0.54) SMN1; SMN2TP53ALDH1A1KMT2ACYP1A2
SCHEMBL6869746 0.87 PLAU (0.43) ADORA2AALDH1A1KMT2ACYP1A2CYP3A4
SCHEMBL6870631 0.86 LMNA (0.48) ADORA2AADORA1TP53ALDH1A1KMT2A
SCHEMBL6872215 0.85 EGLN2 (0.42) SMN1; SMN2ADORA2AADORA1ALDH1A1KMT2A
SCHEMBL6872375 0.84 ADORA2A (0.60) SMN1; SMN2ADORA2AADORA1TP53KMT2A
SCHEMBL6870664 0.82 TP53 (0.45) SMN1; SMN2ADORA2AADORA1TP53ALDH1A1
SCHEMBL6868276 0.82 TP53 (0.44) SMN1; SMN2ADORA2AADORA1TP53ALDH1A1
SCHEMBL6871216 0.82 ADORA2A (0.44) SMN1; SMN2ADORA2AADORA1TP53ALDH1A1
SCHEMBL6870348 0.81 ADORA2A (0.56) SMN1; SMN2ADORA2ATP53ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347974-B1 AMINOTRIAZOLOPYRIDIINE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS HOFFMANN LA ROCHE (CH) 2004-11-03 EP disclosed