SCHEMBL6863739

SCHEMBL6863739

Nc1cc(C(=O)NCc2ccccc2Cl)cc2nc(-c3ccccc3)nn12

nearest known ligand 0.54

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 4/20 0.54
TP53 P04637 5/20 0.46
ALDH1A1 P00352 2/20 0.46
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
GAA P10253 1/20 0.46
TSHR P16473 1/20 0.46
CYP2C19 P33261 1/20 0.46
KMT2A Q03164 1/20 0.46
SCN2A Q99250 1/20 0.46
SCN10A Q9Y5Y9 1/20 0.46
MAPT P10636 3/20 0.46
LMNA P02545 3/20 0.46
HPGD P15428 1/20 0.44
KLKB1 P03952 1/20 0.44
KDM4E B2RXH2 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6863096 0.88 SMN1; SMN2 (0.43) SMN1; SMN2TP53ALDH1A1CYP1A2CYP3A4
SCHEMBL6870074 0.88 KMT2A (0.48) SMN1; SMN2ALDH1A1CYP3A4CYP2C19KMT2A
SCHEMBL6868276 0.87 TP53 (0.44) SMN1; SMN2TP53ALDH1A1CYP1A2CYP3A4
SCHEMBL6867645 0.86 POLB (0.49) SMN1; SMN2TP53ALDH1A1CYP1A2CYP3A4
SCHEMBL6870348 0.86 ADORA2A (0.56) SMN1; SMN2TP53ALDH1A1CYP1A2CYP3A4
SCHEMBL6873157 0.86 HPGDS (0.51) ALDH1A1TSHRCYP2C19LMNAHPGD
SCHEMBL6871254 0.85 ADORA2A (0.56) SMN1; SMN2TP53ALDH1A1CYP1A2CYP3A4
SCHEMBL6872375 0.85 ADORA2A (0.60) SMN1; SMN2TP53KMT2AMAPT
SCHEMBL6870664 0.85 TP53 (0.45) SMN1; SMN2TP53ALDH1A1CYP1A2CYP3A4
SCHEMBL6867448 0.85 HTT (0.56) TP53ALDH1A1GAAKMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347974-B1 AMINOTRIAZOLOPYRIDIINE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS HOFFMANN LA ROCHE (CH) 2004-11-03 EP disclosed