SCHEMBL6871193

SCHEMBL6871193

COc1ccc(-c2nc3cc(C(=O)NCc4ccccc4Br)cc(N)n3n2)s1

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.41
MAPT P10636 2/20 0.40
ALDH1A1 P00352 2/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
ADORA2A P29274 4/20 0.37
PRNP P04156 1/20 0.37
LMNA P02545 1/20 0.36
KDM4E B2RXH2 2/20 0.35
EPHX2 P34913 1/20 0.35
MAPK10 P53779 1/20 0.35
HDAC1 Q13547 1/20 0.35
MEN1 O00255 1/20 0.35
TP53 P04637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6871570 0.90 HPGD (0.46) MAPTALDH1A1CYP3A4LMNAKDM4E
SCHEMBL6869899 0.90 SLC16A3 (0.43) KMT2AMAPTALDH1A1CYP3A4CYP2D6
SCHEMBL6867499 0.89 KMT2A (0.43) KMT2AMAPTALDH1A1CYP3A4CYP2D6
SCHEMBL6863086 0.88 PLAU (0.44) ALDH1A1CYP2D6ADORA2ALMNAKDM4E
SCHEMBL6873046 0.83 ADORA2A (0.56) KMT2AMAPTALDH1A1ADORA2APRNP
SCHEMBL6873034 0.83 ADORA2A (0.39) MAPTALDH1A1ADORA2ALMNAKDM4E
SCHEMBL6872062 0.82 TP53 (0.47) KMT2AMAPTALDH1A1CYP3A4CYP2D6
SCHEMBL6870074 0.81 KMT2A (0.48) KMT2AMAPTALDH1A1CYP3A4ADORA2A
SCHEMBL6867527 0.81 ADORA2A (0.38) KMT2AMAPTALDH1A1ADORA2ALMNA
SCHEMBL6869624 0.81 ADORA2A (0.41) KMT2AMAPTALDH1A1CYP3A4ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347974-B1 AMINOTRIAZOLOPYRIDIINE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS HOFFMANN LA ROCHE (CH) 2004-11-03 EP disclosed