SCHEMBL6863086

SCHEMBL6863086

COc1ccc(-c2nc3cc(C(=O)NCc4ccccc4)cc(N)n3n2)s1

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PLAU P00749 1/20 0.44
CYP2C19 P33261 2/20 0.43
CYP2D6 P10635 1/20 0.42
CHRM4 P08173 1/20 0.42
HPGD P15428 2/20 0.42
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
HSD17B10 Q99714 1/20 0.42
CYP2C9 P11712 1/20 0.41
SCD O00767 2/20 0.41
LMNA P02545 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
HPGDS O60760 1/20 0.41
KLKB1 P03952 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
ADORA2A P29274 2/20 0.40
TP53 P04637 2/20 0.40
CSNK1D P48730 1/20 0.40
CLK1 P49759 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6863351 0.89 PLAU (0.47) PLAUCYP2C19CYP2D6CHRM4HPGD
SCHEMBL6871570 0.88 HPGD (0.46) CYP2C19HPGDKDM4EALDH1A1LMNA
SCHEMBL6869899 0.88 SLC16A3 (0.43) CYP2C19CYP2D6CHRM4HPGDKDM4E
SCHEMBL6871193 0.88 KMT2A (0.41) CYP2D6KDM4EALDH1A1LMNAADORA2A
SCHEMBL6869624 0.86 ADORA2A (0.41) HPGDKDM4EALDH1A1HSD17B10LMNA
SCHEMBL6873034 0.86 ADORA2A (0.39) HPGDKDM4EALDH1A1HSD17B10LMNA
SCHEMBL6867527 0.84 ADORA2A (0.38) HPGDKDM4EALDH1A1LMNASMN1; SMN2
SCHEMBL6870566 0.83 ADORA2A (0.45) CYP2D6HPGDKDM4EALDH1A1LMNA
SCHEMBL6863519 0.83 ADORA2A (0.44) HPGDKDM4EALDH1A1SMN1; SMN2ADORA2A
SCHEMBL6863144 0.83 NAAA (0.39) L3MBTL1ADORA2ATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347974-B1 AMINOTRIAZOLOPYRIDIINE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS HOFFMANN LA ROCHE (CH) 2004-11-03 EP disclosed