SCHEMBL6869899

SCHEMBL6869899

COc1ccc(-c2nc3cc(C(=O)NCc4ccccc4Cl)cc(N)n3n2)s1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC16A3 O15427 1/20 0.43
SLC16A1 P53985 1/20 0.43
MCTS1 Q9ULC4 1/20 0.43
TP53 P04637 2/20 0.42
ALDH1A1 P00352 3/20 0.42
KMT2A Q03164 2/20 0.42
TSHR P16473 2/20 0.42
GAA P10253 2/20 0.42
CYP1A2 P05177 2/20 0.42
CYP3A4 P08684 2/20 0.42
CYP2C19 P33261 2/20 0.42
KLKB1 P03952 1/20 0.42
ROCK2 O75116 2/20 0.42
ROCK1 Q13464 2/20 0.42
MAPT P10636 8/20 0.41
KDM4E B2RXH2 2/20 0.41
CHRM4 P08173 1/20 0.41
LMNA P02545 3/20 0.41
PKM P14618 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6871570 0.90 HPGD (0.46) TP53ALDH1A1GAACYP1A2CYP3A4
SCHEMBL6871193 0.90 KMT2A (0.41) TP53ALDH1A1KMT2ACYP3A4MAPT
SCHEMBL6870466 0.89 TP53 (0.47) TP53ALDH1A1KMT2ATSHRGAA
SCHEMBL6863086 0.88 PLAU (0.44) TP53ALDH1A1CYP2C19KLKB1KDM4E
SCHEMBL6871254 0.83 ADORA2A (0.56) TP53ALDH1A1KMT2ATSHRGAA
SCHEMBL6873034 0.83 ADORA2A (0.39) TP53ALDH1A1GAAMAPTKDM4E
SCHEMBL6872062 0.82 TP53 (0.47) TP53ALDH1A1KMT2AGAACYP1A2
SCHEMBL6863739 0.81 SMN1; SMN2 (0.54) TP53ALDH1A1KMT2ATSHRGAA
SCHEMBL6867527 0.81 ADORA2A (0.38) ALDH1A1KMT2AMAPTKDM4ELMNA
SCHEMBL6869624 0.81 ADORA2A (0.41) TP53ALDH1A1KMT2ATSHRCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347974-B1 AMINOTRIAZOLOPYRIDIINE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS HOFFMANN LA ROCHE (CH) 2004-11-03 EP disclosed