SCHEMBL6872051

SCHEMBL6872051

CC(C)(C)OC(=O)CON(Cc1ccc(F)cc1)C(=O)/C=C(\O)C(=O)O

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NR1D1 P20393 1/20 0.39
RIPK1 Q13546 2/20 0.36
KCNQ4 P56696 3/20 0.35
KCNQ5 Q9NR82 3/20 0.35
KDM1A O60341 2/20 0.34
HDAC8 Q9BY41 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
CTSS P25774 1/20 0.34
CTSK P43235 1/20 0.34
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
MAPT P10636 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6872054 1.00 NR1D1 (0.39) NR1D1RIPK1KCNQ4KCNQ5KDM1A
SCHEMBL6076970 0.90 NR1D1 (0.38) NR1D1RIPK1KCNQ4KCNQ5KDM1A
SCHEMBL6076961 0.90 NR1D1 (0.38) NR1D1RIPK1KCNQ4KCNQ5KDM1A
SCHEMBL6871265 0.84 BCL2A1 (0.36) RIPK1ALDH1A1LMNAMAPTTDP1
SCHEMBL6871267 0.84 BCL2A1 (0.36) RIPK1ALDH1A1LMNAMAPTTDP1
SCHEMBL6881588 0.82 ALDH1A1 (0.40) RIPK1ALDH1A1LMNAMAPTTDP1
SCHEMBL6881585 0.82 ALDH1A1 (0.40) RIPK1ALDH1A1LMNAMAPTTDP1
SCHEMBL6881196 0.82 RIPK1 (0.39) RIPK1ALDH1A1LMNAMAPTTDP1
SCHEMBL6881199 0.82 RIPK1 (0.39) RIPK1ALDH1A1LMNAMAPTTDP1
SCHEMBL3681999 0.79 TDP1 (0.39) RIPK1ALDH1A1LMNAMAPTTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6777440-B2 HIV integrase inhibitors BRISTOL-MYERS SQUIBB COMPANY 2004-08-17 US disclosed
US-20030176495-A1 HIV Integrase inhibitors BRISTOL-MYERS SQUIBB COMPANY 2003-09-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030176495-A1 HIV Integrase inhibitors MAPT, RIF1, HPRT1 NR1D1 955/4885RIPK1 1438/4885KCNQ4 4624/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.