SCHEMBL6872088

SCHEMBL6872088

COc1ccc(CNC(=O)c2cc(N)n3nc(-c4cccs4)nc3c2)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MYC P01106 1/20 0.56
MAX P61244 1/20 0.56
LMNA P02545 5/20 0.54
SMN1; SMN2 Q16637 4/20 0.54
KMT2A Q03164 2/20 0.54
ADORA2A P29274 1/20 0.54
MEN1 O00255 1/20 0.54
ESR1 P03372 1/20 0.54
ALDH1A1 P00352 2/20 0.50
KDM4E B2RXH2 2/20 0.50
HPGD P15428 1/20 0.50
CHRM4 P08173 1/20 0.47
UBE2I P63279 1/20 0.44
SAE1 Q9UBE0 1/20 0.44
UBA2 Q9UBT2 1/20 0.44
POLB P06746 2/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6869924 0.85 CHRM4 (0.47) MYCMAXKMT2AADORA2AMEN1
SCHEMBL6871169 0.82 ADORA2A (0.54) LMNASMN1; SMN2KMT2AADORA2AMEN1
SCHEMBL6870639 0.82 ADORA2A (0.59) SMN1; SMN2ADORA2AALDH1A1UBE2ISAE1
SCHEMBL6870583 0.80 ADORA2A (0.66) SMN1; SMN2KMT2AADORA2AMEN1ALDH1A1
SCHEMBL6870384 0.80 ADORA2A (0.58) LMNASMN1; SMN2ADORA2AALDH1A1KDM4E
SCHEMBL6873589 0.80 ADORA2A (0.56) LMNASMN1; SMN2KMT2AADORA2AMEN1
SCHEMBL6873046 0.80 ADORA2A (0.56) LMNASMN1; SMN2KMT2AADORA2AALDH1A1
SCHEMBL6871254 0.80 ADORA2A (0.56) LMNASMN1; SMN2KMT2AADORA2AALDH1A1
SCHEMBL6873334 0.79 ADORA2A (0.58) ADORA2AALDH1A1HPGDCHRM4NPC1
SCHEMBL6863086 0.79 PLAU (0.44) LMNASMN1; SMN2ADORA2AALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347974-B1 AMINOTRIAZOLOPYRIDIINE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS HOFFMANN LA ROCHE (CH) 2004-11-03 EP disclosed