SCHEMBL6869924

SCHEMBL6869924

COc1ccc(CNC(=O)c2cc(N)n3nc(-c4nccs4)nc3c2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM4 P08173 4/20 0.47
MYC P01106 1/20 0.44
MAX P61244 1/20 0.44
TP53 P04637 1/20 0.43
ALDH1A1 P00352 4/20 0.42
HPGD P15428 3/20 0.42
CYP2C9 P11712 3/20 0.42
KMT2A Q03164 2/20 0.42
CYP1A2 P05177 2/20 0.42
CYP3A4 P08684 2/20 0.42
CYP2C19 P33261 2/20 0.42
KDM1A O60341 1/20 0.42
HDAC1 Q13547 1/20 0.42
HDAC2 Q92769 1/20 0.42
HDAC8 Q9BY41 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
HDAC5 Q9UQL6 1/20 0.42
GAA P10253 1/20 0.42
DHFR P00374 1/20 0.42
KDM4E B2RXH2 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6870516 0.90 KDM4E (0.46) ALDH1A1KMT2AGAADHFRKDM4E
SCHEMBL6867467 0.88 KDM4E (0.46) ALDH1A1HPGDCYP2C9KMT2ACYP1A2
SCHEMBL6873737 0.88 L3MBTL1 (0.43) TP53ALDH1A1HPGDKMT2AHDAC1
SCHEMBL6870625 0.87 MAPK10 (0.45) TP53ALDH1A1CYP2C19GAAKDM4E
SCHEMBL6872088 0.85 MYC (0.56) CHRM4MYCMAXALDH1A1HPGD
SCHEMBL6863441 0.84 HPGD (0.45) TP53ALDH1A1HPGDKMT2ACYP1A2
SCHEMBL6871169 0.83 ADORA2A (0.54) CHRM4KMT2AKDM1AHDAC1HDAC2
SCHEMBL6871432 0.83 ADORA2A (0.40) TP53ALDH1A1HPGDKMT2AHDAC2
SCHEMBL6867623 0.80 F2 (0.43) ALDH1A1HPGDKMT2AHDAC1HDAC6
SCHEMBL6872077 0.80 ADORA2A (0.42) ALDH1A1HPGDKMT2ADHFRKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347974-B1 AMINOTRIAZOLOPYRIDIINE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS HOFFMANN LA ROCHE (CH) 2004-11-03 EP disclosed