SCHEMBL6872109

SCHEMBL6872109

Cc1c(C)c(C)c(CNC2CCC(Nc3nccc(N(C)C)n3)CC2)c(C)c1C

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 2/20 0.36
BACE1 P56817 1/20 0.36
MCHR1 Q99705 7/20 0.36
ADRA2A P08913 3/20 0.36
HRH1 P35367 3/20 0.36
HTR2B P41595 3/20 0.36
ADRA1A P35348 1/20 0.36
MAPK8 P45983 2/20 0.36
MAPK9 P45984 2/20 0.36
MAPK10 P53779 2/20 0.36
CDK4 P11802 3/20 0.36
CDK1 P06493 2/20 0.36
CCNB1 P14635 2/20 0.36
CCNA2 P20248 2/20 0.36
CCND1 P24385 2/20 0.36
CDK2 P24941 2/20 0.36
CCNA1 P78396 2/20 0.36
CTSK P43235 1/20 0.35
HRH4 Q9H3N8 2/20 0.35
MAPK14 Q16539 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6877522 1.00 ACHE (0.36) ACHEBACE1MCHR1ADRA2AHRH1
SCHEMBL6875559 0.86 MCHR1 (0.42) MCHR1ADRA2AHRH1HTR2BADRA1A
SCHEMBL6879311 0.83 MAPK8 (0.43) ACHEBACE1MCHR1ADRA2AMAPK8
SCHEMBL6879316 0.83 MAPK8 (0.43) ACHEBACE1MCHR1ADRA2AMAPK8
SCHEMBL6875096 0.81 MCHR1 (0.37) ACHEBACE1MCHR1ADRA2AHRH1
SCHEMBL6875101 0.81 MCHR1 (0.37) ACHEBACE1MCHR1ADRA2AHRH1
SCHEMBL6873935 0.79 ACHE (0.38) ACHEBACE1MAPK8MAPK9MAPK10
SCHEMBL6873931 0.79 ACHE (0.38) ACHEBACE1MAPK8MAPK9MAPK10
SCHEMBL6464494 0.79 CTSK (0.41) MCHR1ADRA2AHRH1HTR2BADRA1A
SCHEMBL6873078 0.78 TSHR (0.51) ACHEBACE1MCHR1ADRA2AMERTK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1464335-A2 Quinoline, tetrahydroquinoline and pyrimidine derivatives as mch antagonist Taisho Pharmaceutical Co. Ltd. (JP) 2004-10-06 EP disclosed