SCHEMBL6874008

SCHEMBL6874008

Cc1cc(NC2CCC(NC(=O)Nc3cccc(Oc4ccccc4)c3)CC2)nc2ccccc12

nearest known ligand 0.53

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.53
KDM4E B2RXH2 1/20 0.53
LMNA P02545 1/20 0.53
USP30 Q70CQ3 2/20 0.49
NPC1 O15118 4/20 0.47
RAB9A P51151 3/20 0.47
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
POLB P06746 1/20 0.47
MAPT P10636 1/20 0.47
EPHX1 P07099 1/20 0.47
TP53 P04637 1/20 0.44
IDH1 O75874 1/20 0.43
EPHX2 P34913 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6874005 1.00 SMN1; SMN2 (0.53) SMN1; SMN2KDM4ELMNAUSP30NPC1
SCHEMBL6877349 0.92 EPHX1 (0.56) SMN1; SMN2KDM4ELMNARAB9AMEN1
SCHEMBL6877352 0.92 EPHX1 (0.56) SMN1; SMN2KDM4ELMNARAB9AMEN1
Trifluoroacetic Acid SCHEMBL6457766 0.88 NPC1 (0.52) SMN1; SMN2KDM4ELMNANPC1RAB9A
SCHEMBL6873829 0.87 LMNA (0.53) SMN1; SMN2KDM4ELMNAMEN1KMT2A
SCHEMBL6873823 0.87 LMNA (0.53) SMN1; SMN2KDM4ELMNAMEN1KMT2A
Trifluoroacetic Acid SCHEMBL6458355 0.82 LMNA (0.49) SMN1; SMN2KDM4ELMNANPC1RAB9A
SCHEMBL6877589 0.80 EPHX1 (0.53) MAPTEPHX1EPHX2
Trifluoroacetic Acid SCHEMBL6457569 0.79 KDM4E (0.52) SMN1; SMN2KDM4ELMNAEPHX1
Trifluoroacetic Acid SCHEMBL6461174 0.78 SMN1; SMN2 (0.49) SMN1; SMN2KDM4ELMNANPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1464335-A2 Quinoline, tetrahydroquinoline and pyrimidine derivatives as mch antagonist Taisho Pharmaceutical Co. Ltd. (JP) 2004-10-06 EP disclosed