SCHEMBL6874231

SCHEMBL6874231

CCCN(CC1CC1)C(=O)Oc1cc(N)n2nc(-c3ccccn3)nc2c1

nearest known ligand 0.48

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 4/20 0.48
F12 P00748 6/20 0.38
F2 P00734 4/20 0.38
CRHR1 P34998 5/20 0.37
HCRTR1 O43613 1/20 0.36
HCRTR2 O43614 1/20 0.36
PLAU P00749 1/20 0.35
KLKB1 P03952 1/20 0.35
HTR1A P08908 1/20 0.35
HTR2A P28223 1/20 0.35
SLC6A9 P48067 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6869475 0.86 ADORA2A (0.55) ADORA2AF12F2CRHR1HCRTR1
SCHEMBL6874003 0.81 ADORA2A (0.59) ADORA2A
SCHEMBL6867998 0.81 ADORA2A (0.52) ADORA2AF12F2PLAUKLKB1
SCHEMBL6867654 0.80 ADORA2A (0.51) ADORA2AF12F2PLAU
SCHEMBL6871499 0.80 ADORA2A (0.47) ADORA2AF12F2PLAUKLKB1
SCHEMBL6867223 0.78 ADORA2A (0.60) ADORA2AF12F2PLAUKLKB1
SCHEMBL6872444 0.75 ADORA2A (0.48) ADORA2AF12F2PLAUKLKB1
SCHEMBL6869823 0.75 ADORA2A (0.56) ADORA2AF12F2PLAUHTR1A
SCHEMBL6871898 0.74 ADORA2A (0.62) ADORA2AF12F2PLAUKLKB1
SCHEMBL6873153 0.73 ADORA2A (0.38) ADORA2AF2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347974-B1 AMINOTRIAZOLOPYRIDIINE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS HOFFMANN LA ROCHE (CH) 2004-11-03 EP claimed