SCHEMBL6874530

SCHEMBL6874530

CN(C)c1nc(N[C@H]2CC[C@@H](NC(=O)Nc3cccc(C(F)(F)F)c3F)CC2)nc2c1CCCC2

nearest known ligand 0.56

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 2/20 0.56
MCHR1 Q99705 15/20 0.42
ADRA2A P08913 11/20 0.42
HRH1 P35367 4/20 0.40
HTR2B P41595 4/20 0.40
ADRA1A P35348 3/20 0.40
HTR1A P08908 1/20 0.39
NPY5R Q15761 1/20 0.39
GAA P10253 1/20 0.38
TP53 P04637 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6874535 1.00 EPHX2 (0.56) EPHX2MCHR1ADRA2AHRH1HTR2B
SCHEMBL6875871 0.92 EPHX2 (0.45) EPHX2MCHR1ADRA2AHRH1HTR2B
SCHEMBL6875875 0.92 EPHX2 (0.45) EPHX2MCHR1ADRA2AHRH1HTR2B
SCHEMBL6875410 0.86 MCHR1 (0.51) MCHR1ADRA2AHRH1HTR2BADRA1A
SCHEMBL6875414 0.86 MCHR1 (0.51) MCHR1ADRA2AHRH1HTR2BADRA1A
SCHEMBL6876354 0.86 P2RY1 (0.44) MCHR1ADRA2AHRH1HTR2BADRA1A
SCHEMBL6876347 0.86 P2RY1 (0.44) MCHR1ADRA2AHRH1HTR2BADRA1A
SCHEMBL6869030 0.86 KMT2A (0.52) EPHX2MCHR1ADRA2AHRH1HTR2B
SCHEMBL6869037 0.86 KMT2A (0.52) EPHX2MCHR1ADRA2AHRH1HTR2B
SCHEMBL6874772 0.84 MCHR1 (0.44) MCHR1ADRA2AHRH1HTR2BADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1464335-A2 Quinoline, tetrahydroquinoline and pyrimidine derivatives as mch antagonist Taisho Pharmaceutical Co. Ltd. (JP) 2004-10-06 EP disclosed