SCHEMBL6875844

SCHEMBL6875844

COc1ccc(CNC2CCC(Nc3ncc(C)c(N(C)C)n3)CC2)cc1C

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 12/20 0.48
ADRA2A P08913 7/20 0.48
HTR2B P41595 6/20 0.48
HRH1 P35367 5/20 0.48
ADRA1A P35348 4/20 0.48
HTR1A P08908 1/20 0.44
KDM1A O60341 1/20 0.41
MAOA P21397 1/20 0.41
MAOB P27338 1/20 0.41
ACHE P22303 2/20 0.41
APP P05067 1/20 0.41
BCHE P06276 1/20 0.41
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
SUV39H2 Q9H5I1 1/20 0.38
PDE5A O76074 1/20 0.37
MAPK8 P45983 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6875836 1.00 MCHR1 (0.48) MCHR1ADRA2AHTR2BHRH1ADRA1A
SCHEMBL6464429 0.85 TSHR (0.50) MCHR1ADRA2AHTR2BHRH1ADRA1A
SCHEMBL6877606 0.85 TSHR (0.50) MCHR1ADRA2AHTR2BHRH1ADRA1A
SCHEMBL6879245 0.84 MCHR1 (0.63) MCHR1ADRA2AHTR2BHRH1ADRA1A
SCHEMBL6879241 0.84 MCHR1 (0.63) MCHR1ADRA2AHTR2BHRH1ADRA1A
Trifluoroacetic Acid SCHEMBL6458250 0.84 MCHR1 (0.47) MCHR1ADRA2AHTR2BHRH1ADRA1A
SCHEMBL6875990 0.84 MCHR1 (0.63) MCHR1ADRA2AHTR2BHRH1ADRA1A
SCHEMBL6875998 0.84 MCHR1 (0.63) MCHR1ADRA2AHTR2BHRH1ADRA1A
SCHEMBL6875146 0.84 MCHR1 (0.53) MCHR1ADRA2AHTR2BHRH1ADRA1A
SCHEMBL6875152 0.84 MCHR1 (0.53) MCHR1ADRA2AHTR2BHRH1ADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1464335-A2 Quinoline, tetrahydroquinoline and pyrimidine derivatives as mch antagonist Taisho Pharmaceutical Co. Ltd. (JP) 2004-10-06 EP disclosed