SCHEMBL6876228

SCHEMBL6876228

[CH2]C#Cc1ccc(-c2ncc(Br)cn2)cc1

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 6/20 0.42
RAB9A P51151 6/20 0.42
SMN1; SMN2 Q16637 4/20 0.42
NFKB1 P19838 2/20 0.42
NFKB2 Q00653 2/20 0.42
RELA Q04206 2/20 0.42
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
KDM4E B2RXH2 2/20 0.34
HSD17B10 Q99714 2/20 0.34
ALDH1A1 P00352 1/20 0.34
TP53 P04637 1/20 0.34
MAPT P10636 1/20 0.34
HPGD P15428 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6847737 0.81 HDAC4 (0.35) NPC1RAB9ASMN1; SMN2NFKB1NFKB2
SCHEMBL6854012 0.79 CLK4 (0.44) NPC1RAB9ASMN1; SMN2NFKB1NFKB2
SCHEMBL6869984 0.77 ALDH1A1 (0.43) NPC1RAB9ASMN1; SMN2NFKB1NFKB2
SCHEMBL6850629 0.77 RAB9A (0.37) NPC1RAB9ASMN1; SMN2MEN1KMT2A
SCHEMBL6881921 0.77 NPC1 (0.39) NPC1RAB9ASMN1; SMN2NFKB1NFKB2
SCHEMBL17629994 0.77 NPC1 (0.44) NPC1RAB9ASMN1; SMN2NFKB1NFKB2
SCHEMBL16222829 0.75 NPC1 (0.65) NPC1RAB9ASMN1; SMN2NFKB1NFKB2
SCHEMBL6852551 0.73 NPC1 (0.54) NPC1RAB9ASMN1; SMN2NFKB1NFKB2
SCHEMBL20488929 0.73 CYP2A6 (0.44) MEN1KMT2AKDM4EALDH1A1
SCHEMBL7466728 0.70 NPC1 (0.48) NPC1RAB9ASMN1; SMN2NFKB1NFKB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1585775-A 6-O-acyl ketolide derivatives of erythromycine useful as antibacterials ORTHO MCNEIL PHARM INC (US) 2005-02-23 CN disclosed
US-6825170-B2 ERYTHROMYCIN TYPE MACROLIDE WITH A FUSED OXAZOLONE RING ORTHO-MCNEIL PHARMACEUTICAL, INC. 2004-11-30 US disclosed