SCHEMBL6876231

SCHEMBL6876231

COc1ccccc1CC(=O)NCCC(N)=O

nearest known ligand 0.67

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 1/20 0.67
NPSR1 Q6W5P4 2/20 0.61
ALDH1A1 P00352 2/20 0.59
HSD17B10 Q99714 1/20 0.59
MEN1 O00255 2/20 0.58
KMT2A Q03164 2/20 0.58
NPC1 O15118 1/20 0.58
RAB9A P51151 1/20 0.58
POLB P06746 1/20 0.56
BCHE P06276 1/20 0.55
CHRM2 P08172 1/20 0.55
ACHE P22303 1/20 0.55
MAPT P10636 1/20 0.53
TSHR P16473 1/20 0.53
MAPK8 P45983 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3205671 0.87 TAAR1 (0.72) TAAR1NPSR1ALDH1A1HSD17B10MEN1
SCHEMBL5843237 0.81 MAPK8 (0.50) ALDH1A1MEN1KMT2ANPC1RAB9A
SCHEMBL22170167 0.80 TAAR1 (0.67) TAAR1NPSR1ALDH1A1HSD17B10MEN1
SCHEMBL1010680 0.80 LMNA (0.64) TAAR1MEN1KMT2APOLBMAPT
SCHEMBL3993600 0.79 NPSR1 (0.79) TAAR1NPSR1BCHECHRM2ACHE
SCHEMBL2826584 0.79 GAA (0.64) TAAR1ALDH1A1MEN1KMT2ANPC1
SCHEMBL29907950 0.79 GAA (0.64) TAAR1ALDH1A1MEN1KMT2ANPC1
SCHEMBL1520822 0.79 NPSR1 (0.68) NPSR1ALDH1A1MEN1KMT2ANPC1
SCHEMBL28465013 0.78 NPC1 (0.81) TAAR1NPSR1ALDH1A1MEN1KMT2A
SCHEMBL9447512 0.78 CA12 (0.65) TAAR1NPSR1BCHECHRM2ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1452522-A2 Novel compounds and compositions as protease inhibitors AXYS PHARMACEUTICALS, INC. (US) 2004-09-01 EP disclosed