SCHEMBL6876456

SCHEMBL6876456

CC(C)(C)C(NC(=O)c1cc2ccccc2[nH]1)C(=O)N1CCN(C(=O)c2nc3ccccc3[nH]2)CC1

nearest known ligand 0.53

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 8/20 0.53
CYP51A1 Q16850 1/20 0.45
SMYD3 Q9H7B4 1/20 0.45
DRD3 P35462 2/20 0.43
DRD2 P14416 2/20 0.43
RBP4 P02753 1/20 0.43
AKR1C3 P42330 2/20 0.43
HRH3 Q9Y5N1 1/20 0.43
HDAC6 Q9UBN7 1/20 0.42
POLB P06746 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
PDE10A Q9Y233 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2227969 0.88 HRH4 (0.45) HRH4CYP51A1SMYD3DRD2RBP4
SCHEMBL6873804 0.88 HRH4 (0.43) HRH4CYP51A1SMYD3DRD2AKR1C3
SCHEMBL2227562 0.84 DRD2 (0.42) HRH4CYP51A1SMYD3DRD2AKR1C3
SCHEMBL1550512 0.83 DRD2 (0.42) HRH4CYP51A1SMYD3DRD2PDE10A
SCHEMBL1550154 0.77 HRH4 (0.38) HRH4SMYD3DRD2SMN1; SMN2PDE10A
SCHEMBL1550169 0.77 ALOX15 (0.44) HRH4CYP51A1SMYD3HRH3PDE10A
SCHEMBL1550577 0.77 TP53 (0.39) HRH4SMYD3DRD2AKR1C3POLB
SCHEMBL1550827 0.77 PYGL (0.44) CYP51A1SMYD3
SCHEMBL1550291 0.76 CYP51A1 (0.42) HRH4CYP51A1SMYD3HRH3PDE10A
SCHEMBL1549798 0.76 AR (0.42) HRH4CYP51A1SMYD3DRD2HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011091410-A1 TRPV4 ANTAGONISTS GLAXOS SMITHKLINE LLC (US) 2011-07-28 WO disclosed