SCHEMBL6877480

SCHEMBL6877480

CN(C)c1nc(NC2CCC(NC(=O)Nc3ccc(OCc4ccccc4)cc3)CC2)nc2c1CCCC2

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NOX1 Q9Y5S8 2/20 0.48
GBA1 P04062 1/20 0.43
RAB9A P51151 3/20 0.43
NPC1 O15118 2/20 0.43
MEN1 O00255 5/20 0.42
KMT2A Q03164 5/20 0.42
PABPC1 P11940 1/20 0.42
ADRA2A P08913 1/20 0.41
MCHR1 Q99705 1/20 0.41
EPHX1 P07099 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
DHODH Q02127 1/20 0.41
S1PR1 P21453 1/20 0.41
OPRM1 P35372 1/20 0.41
OPRD1 P41143 1/20 0.41
LTA4H P09960 1/20 0.40
FAAH O00519 1/20 0.40
EPHX2 P34913 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6877475 1.00 NOX1 (0.48) NOX1GBA1RAB9ANPC1MEN1
SCHEMBL6876429 0.90 USP30 (0.43) RAB9ANPC1KMT2AADRA2AMCHR1
SCHEMBL6876423 0.90 USP30 (0.43) RAB9ANPC1KMT2AADRA2AMCHR1
SCHEMBL6866751 0.89 NPC1 (0.56) RAB9ANPC1MEN1KMT2AEPHX1
SCHEMBL6866756 0.89 NPC1 (0.56) RAB9ANPC1MEN1KMT2AEPHX1
SCHEMBL6874492 0.89 EPHX1 (0.54) RAB9ANPC1ADRA2AMCHR1EPHX1
SCHEMBL6874485 0.89 EPHX1 (0.54) RAB9ANPC1ADRA2AMCHR1EPHX1
SCHEMBL6876164 0.87 NPC1 (0.47) RAB9ANPC1MEN1KMT2AADRA2A
SCHEMBL6876167 0.87 NPC1 (0.47) RAB9ANPC1MEN1KMT2AADRA2A
SCHEMBL6874504 0.86 MCHR1 (0.44) RAB9AADRA2AMCHR1EPHX1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1464335-A2 Quinoline, tetrahydroquinoline and pyrimidine derivatives as mch antagonist Taisho Pharmaceutical Co. Ltd. (JP) 2004-10-06 EP disclosed