SCHEMBL6876164

SCHEMBL6876164

CCCCOc1ccc(NC(=O)N[C@H]2CC[C@@H](Nc3nc4c(c(N(C)C)n3)CCCC4)CC2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.47
RAB9A P51151 3/20 0.47
EPHX2 P34913 3/20 0.45
EPHX1 P07099 3/20 0.45
AURKA O14965 2/20 0.42
AURKB Q96GD4 2/20 0.42
MAPT P10636 2/20 0.41
TP53 P04637 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
HDAC1 Q13547 3/20 0.41
HDAC8 Q9BY41 3/20 0.41
HDAC6 Q9UBN7 3/20 0.41
MEN1 O00255 1/20 0.40
POLB P06746 1/20 0.40
KMT2A Q03164 1/20 0.40
JAK2 O60674 1/20 0.40
ADRA2A P08913 1/20 0.39
HRH1 P35367 1/20 0.39
HTR2B P41595 1/20 0.39
MCHR1 Q99705 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6876167 1.00 NPC1 (0.47) NPC1RAB9AEPHX2EPHX1AURKA
SCHEMBL6876601 0.98 EPHX2 (0.46) NPC1RAB9AEPHX2EPHX1AURKA
SCHEMBL6876610 0.98 EPHX2 (0.46) NPC1RAB9AEPHX2EPHX1AURKA
SCHEMBL6866756 0.93 NPC1 (0.56) NPC1RAB9AEPHX2EPHX1MAPT
SCHEMBL6866751 0.93 NPC1 (0.56) NPC1RAB9AEPHX2EPHX1MAPT
SCHEMBL6877142 0.90 RAB9A (0.47) NPC1RAB9AEPHX2EPHX1MAPT
SCHEMBL6877139 0.90 RAB9A (0.47) NPC1RAB9AEPHX2EPHX1MAPT
SCHEMBL6879538 0.90 EPHX1 (0.56) NPC1RAB9AEPHX2EPHX1AURKB
SCHEMBL6879546 0.90 EPHX1 (0.56) NPC1RAB9AEPHX2EPHX1AURKB
SCHEMBL6874878 0.88 NPC1 (0.54) NPC1RAB9AEPHX2EPHX1AURKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1464335-A2 Quinoline, tetrahydroquinoline and pyrimidine derivatives as mch antagonist Taisho Pharmaceutical Co. Ltd. (JP) 2004-10-06 EP disclosed