SCHEMBL687797

SCHEMBL687797

CCOC(=O)OC1=CN(C(=O)c2sc(-c3ccccc3)nc2C)CCc2c1[nH]c1ccccc21

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 4/20 0.46
CNR1 P21554 1/20 0.42
CDC7 O00311 3/20 0.41
DBF4 Q9UBU7 3/20 0.41
TRPM8 Q7Z2W7 1/20 0.41
ALOX5 P09917 1/20 0.40
HPGD P15428 3/20 0.39
NPC1 O15118 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
ALDH1A1 P00352 4/20 0.38
MAPT P10636 3/20 0.38
KMT2A Q03164 2/20 0.38
CYP1A2 P05177 2/20 0.38
AURKA O14965 1/20 0.38
MAPK10 P53779 1/20 0.38
RIPK1 Q13546 1/20 0.38
MEN1 O00255 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL715227 0.87 CDC7 (0.43) NR1H4CDC7DBF4NPC1SMN1; SMN2
SCHEMBL273588 0.87 NR1H4 (0.62) NR1H4CNR1CDC7DBF4TRPM8
SCHEMBL688979 0.86 NR1H4 (0.47) NR1H4ALOX5HPGDNPC1SMN1; SMN2
SCHEMBL688779 0.78 NR1H4 (0.45) NR1H4ALDH1A1MAPTKMT2AAURKA
SCHEMBL275094 0.74 NR1H4 (0.57) NR1H4CDC7DBF4NPC1ALDH1A1
SCHEMBL274417 0.74 NR1H4 (0.62) NR1H4HPGDNPC1ALDH1A1MAPT
SCHEMBL687997 0.74 NR1H4 (0.53) NR1H4HPGDNPC1SMN1; SMN2ALDH1A1
SCHEMBL687825 0.74 NR1H4 (0.53) NR1H4HPGDNPC1SMN1; SMN2ALDH1A1
SCHEMBL274293 0.69 NR1H4 (0.65) NR1H4HPGDALDH1A1MAPTKMT2A
SCHEMBL688726 0.69 BAZ2B (0.40) NR1H4HPGDNPC1SMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1532153-B1 AZEPINOINDOLE AND PYRIDOINDOLE DERIVATIVES AS PHARMACEUTICAL AGENTS X CEPTOR THERAPEUTICS INC (US) 2012-02-29 EP claimed