SCHEMBL6878307

SCHEMBL6878307

COc1ccc(CN[C@H]2CC[C@@H](Nc3nccc(N(C)C)n3)CC2)c(OC)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 9/20 0.46
CYP1A2 P05177 9/20 0.46
CYP3A4 P08684 9/20 0.46
CYP2D6 P10635 8/20 0.46
CYP2C19 P33261 8/20 0.46
USP2 O75604 7/20 0.46
HSD17B10 Q99714 4/20 0.46
LMNA P02545 3/20 0.46
ALDH1A1 P00352 3/20 0.46
CASP7 P55210 1/20 0.46
APLNR P35414 1/20 0.42
FLT3 P36888 1/20 0.42
TYRO3 Q06418 1/20 0.42
MERTK Q12866 1/20 0.42
GAS6 Q14393 1/20 0.42
KMT2A Q03164 6/20 0.41
MEN1 O00255 5/20 0.41
CLK4 Q9HAZ1 2/20 0.41
MCHR1 Q99705 2/20 0.41
ACHE P22303 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6878316 1.00 TSHR (0.46) TSHRCYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL6877439 0.89 ACHE (0.42) ALDH1A1KMT2AMEN1MCHR1ACHE
SCHEMBL6877433 0.89 ACHE (0.42) ALDH1A1KMT2AMEN1MCHR1ACHE
SCHEMBL6874596 0.88 APLNR (0.44) TSHRCYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL6459873 0.88 APLNR (0.44) TSHRCYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL6875945 0.84 ACHE (0.41) TSHRHSD17B10ALDH1A1KMT2AMEN1
SCHEMBL6875957 0.84 ACHE (0.41) TSHRHSD17B10ALDH1A1KMT2AMEN1
SCHEMBL6873081 0.84 TSHR (0.51) TSHRALDH1A1FLT3TYRO3MERTK
SCHEMBL6873078 0.84 TSHR (0.51) TSHRALDH1A1FLT3TYRO3MERTK
SCHEMBL6875163 0.84 EIF2AK2 (0.46) CYP1A2CYP3A4CYP2D6CYP2C19USP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1464335-A2 Quinoline, tetrahydroquinoline and pyrimidine derivatives as mch antagonist Taisho Pharmaceutical Co. Ltd. (JP) 2004-10-06 EP disclosed