SCHEMBL6878366

SCHEMBL6878366

O=C(O)Cc1csc(NC(=O)CNC23CC4CCCC(C2)C(C4)C3)n1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
ALDH1A1 P00352 3/20 0.38
ITGB1 P05556 1/20 0.38
ITGA4 P13612 1/20 0.38
PDE5A O76074 5/20 0.37
KDM4E B2RXH2 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
CNR1 P21554 1/20 0.36
CNR2 P34972 1/20 0.36
HTT P42858 2/20 0.36
NPC1 O15118 1/20 0.36
LMNA P02545 1/20 0.36
RAB9A P51151 1/20 0.36
POLB P06746 1/20 0.36
GAA P10253 1/20 0.36
OGFRL1 Q5TC84 1/20 0.36
PDE1A P54750 1/20 0.35
PDE1B Q01064 1/20 0.35
PDE1C Q14123 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6878139 0.77 PDE5A (0.47) MEN1KMT2APDE5AKDM4EPDE1A
SCHEMBL6879293 0.72 GAA (0.49) ALDH1A1TDP1CNR2HTTNPC1
SCHEMBL6876782 0.72 PDE5A (0.42) PDE5AKDM4EPDE1APDE1BPDE1C
SCHEMBL1758817 0.70 PDE5A (0.50) MEN1KMT2APDE5AKDM4EPDE1A
SCHEMBL6880848 0.70 PDE5A (0.41) PDE5AKDM4EPDE1APDE1BPDE1C
SCHEMBL7488591 0.69 KMT2A (0.53) MEN1KMT2AALDH1A1ITGB1ITGA4
SCHEMBL1758662 0.68 EPHX2 (0.49) KMT2AALDH1A1TDP1CNR2HTT
SCHEMBL6036808 0.66 ALDH1A1 (0.54) MEN1KMT2AALDH1A1ITGB1ITGA4
SCHEMBL8350301 0.66 ALDH1A1 (0.54) MEN1KMT2AALDH1A1ITGB1ITGA4
SCHEMBL7493963 0.66 ALDH1A1 (0.54) MEN1KMT2AALDH1A1ITGB1ITGA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011058582-A1 HISTONE DEACETYLASE INHIBITORS FOR THE TREATMENT OF FUNGAL INFECTIONS ORCHID RESEARCH LABORATORIES LTD. (IN) 2011-05-19 WO disclosed