SCHEMBL6879124

SCHEMBL6879124

Nc1ccc(-n2cnc3ncncc32)c2ccccc12

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 2/20 0.40
CYP17A1 P05093 1/20 0.36
LTA4H P09960 1/20 0.35
PI4KA P42356 1/20 0.34
PI4K2B Q8TCG2 1/20 0.34
PI4K2A Q9BTU6 1/20 0.34
PI4KB Q9UBF8 1/20 0.34
HDAC1 Q13547 1/20 0.31
HDAC3 O15379 1/20 0.31
IDO1 P14902 1/20 0.31
EP300 Q09472 1/20 0.31
KAT2B Q92831 1/20 0.31
KAT8 Q9H7Z6 1/20 0.31
NCOR2 Q9Y618 1/20 0.31
HCAR1 Q9BXC0 1/20 0.30
ALDH1A1 P00352 1/20 0.30
HTT P42858 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6638826 0.79 CTSB (0.46) HDAC6ALDH1A1HTT
SCHEMBL6872767 0.78 PI4KA (0.42) LTA4HPI4KAPI4K2BPI4K2API4KB
SCHEMBL6667117 0.75 FGFR1 (0.56) CYP17A1LTA4HHCAR1ALDH1A1HTT
SCHEMBL6664459 0.72 HDAC6 (0.58) HDAC6LTA4HALDH1A1HTT
SCHEMBL6661764 0.67 HDAC6 (0.59) HDAC6CYP17A1LTA4HHDAC1HCAR1
SCHEMBL2010867 0.66 HDAC6 (0.43) HDAC6LTA4HHDAC1
SCHEMBL6664883 0.65 CDC7 (0.49) HTT
SCHEMBL8327824 0.64 HDAC6 (0.59) HDAC6CYP17A1LTA4HHDAC1ALDH1A1
SCHEMBL2623743 0.63 HDAC6 (0.44) HDAC6LTA4HHDAC1
SCHEMBL8326090 0.63 HDAC6 (0.58) HDAC6KAT2BALDH1A1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6825184-B2 FOR USE AS ANTI-INFLAMMATORY AGENTS BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. 2004-11-30 US disclosed
US-20030162968-A1 1,4-Disubstituted benzo-fused urea compounds BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. 2003-08-28 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030162968-A1 1,4-Disubstituted benzo-fused urea compounds NFKBIA, MPO, RELA HDAC6 219/4885CYP17A1 1310/4885LTA4H 329/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.