SCHEMBL687934

SCHEMBL687934

Cc1ccc([C@H](CC(=O)O)NC(=O)Nc2cc(C(F)(F)F)cn(Cc3ccccc3)c2=O)cc1

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.47
CYP2C9 P11712 2/20 0.43
CYP2C19 P33261 2/20 0.43
KDM4E B2RXH2 1/20 0.43
MEN1 O00255 1/20 0.43
ALDH1A1 P00352 1/20 0.43
HPGD P15428 1/20 0.43
CTSA P10619 3/20 0.42
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
MAPT P10636 1/20 0.41
ITGB1 P05556 4/20 0.41
ITGA4 P13612 4/20 0.41
POLB P06746 1/20 0.40
MCHR1 Q99705 1/20 0.40
TP53 P04637 1/20 0.40
PTGER3 P43115 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL687707 0.79 PTGER3 (0.58) KMT2AKDM4EALDH1A1CTSAMAPT
SCHEMBL688469 0.78 KDM4E (0.58) KMT2ACYP2C9CYP2C19KDM4EMEN1
SCHEMBL688126 0.78 KDM4E (0.56) KMT2ACYP2C9CYP2C19KDM4EMEN1
SCHEMBL687488 0.77 MAPT (0.51) KMT2AKDM4EMEN1ALDH1A1CTSA
SCHEMBL687985 0.77 KDM4E (0.46) KMT2ACYP2C9CYP2C19KDM4EMEN1
SCHEMBL687613 0.77 PTGER3 (0.55) KMT2ACYP2C9CYP2C19KDM4EMEN1
SCHEMBL687952 0.76 PTGER3 (0.51) KMT2ACYP2C9CYP2C19KDM4EMEN1
SCHEMBL688082 0.76 TP53 (0.41) KMT2AKDM4EMEN1ALDH1A1CTSA
SCHEMBL687856 0.76 ALDH1A1 (0.58) KMT2ACYP2C9CYP2C19KDM4EMEN1
SCHEMBL688231 0.76 KDM4E (0.53) KMT2ACYP2C9CYP2C19KDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1203766-B1 Carboxylic acid derivatives that inhibit the binding of integrins to their receptors ENCYSIVE PHARMACEUTICALS INC (US) 2012-02-29 EP disclosed
EP-1203766-A2 Carboxylic acid derivatives that inhibit the binding of integrins to their receptors TEXAS BIOTECHNOLOGY CORPORATION (US) 2002-05-08 EP disclosed