SCHEMBL687973

SCHEMBL687973

CCOC(=O)/C=C/CP(=O)(OCC)OCC

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.47
HCAR2 Q8TDS4 1/20 0.47
ALDH1A1 P00352 1/20 0.42
TSHR P16473 1/20 0.40
PPARD Q03181 1/20 0.39
TTR P02766 1/20 0.38
DPP4 P27487 1/20 0.38
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA7 P43166 1/20 0.38
CA9 Q16790 1/20 0.38
CA14 Q9ULX7 1/20 0.38
NPSR1 Q6W5P4 1/20 0.37
CYP3A4 P08684 1/20 0.36
HTT P42858 1/20 0.35
RAB9A P51151 1/20 0.35
ATM Q13315 1/20 0.34
LMNA P02545 1/20 0.33
MDM2 Q00987 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1399032 1.00 MAPT (0.47) MAPTHCAR2ALDH1A1TSHRPPARD
Butyric Acid SCHEMBL11237541 0.89 HCAR2 (0.42) MAPTHCAR2ALDH1A1TSHRPPARD
SCHEMBL17398721 0.88 MAPT (0.42) MAPTHCAR2ALDH1A1TSHRPPARD
SCHEMBL6231924 0.85 HCAR2 (0.43) MAPTHCAR2TSHRPPARDTTR
SCHEMBL4978281 0.85 HCAR2 (0.43) MAPTHCAR2TSHRPPARDTTR
SCHEMBL13502893 0.85 MAPT (0.47) MAPTHCAR2ALDH1A1TSHRTTR
SCHEMBL6382885 0.85 NPSR1 (0.40) MAPTHCAR2ALDH1A1TSHRPPARD
SCHEMBL6382879 0.85 NPSR1 (0.40) MAPTHCAR2ALDH1A1TSHRPPARD
SCHEMBL8620959 0.84 MAPT (0.46) MAPTHCAR2ALDH1A1PPARDTTR
SCHEMBL15163745 0.84 MAPT (0.46) MAPTHCAR2ALDH1A1TSHRTTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 474 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2644612-B1 Method for producing sanshool TSUMURA & CO (JP) 2016-01-06 EP claimed
US-8877953-B2 Method for producing sanshool TSUMURA & CO. (JP) 2014-11-04 US claimed
US-20130261327-A1 METHOD FOR PRODUCING SANSHOOL TSUMURA & CO. (JP) 2013-10-03 US claimed
EP-2644612-A1 Method for producing sanshool TSUMURA & CO. (JP) 2013-10-02 EP claimed
JP-62129246-A None JP disclosed
US-20260116838-A1 NEOCARZILIN DERIVATIVES AS ANTIMETASTATIC AGENTS PURDUE RESEARCH FOUNDATION (US) 2026-04-30 US disclosed
US-12570672-B2 Macrocyclic compounds and methods of use AMGEN INC. 2026-03-10 US disclosed
WO-2025262297-A1 PROTAC DEGRADERS OF MLLT1 AND/OR MLLT3 DARK BLUE THERAPEUTICS LTD (GB) 2025-12-26 WO disclosed
WO-2025262295-A1 PROTAC DEGRADERS OF MLLT1 AND/OR MLLT3 DARK BLUE THERAPEUTICS LTD (GB) 2025-12-26 WO disclosed
EP-4667466-A1 PROTAC DEGRADERS OF MLLT1 AND/OR MLLT3 Dark Blue Therapeutics Ltd (GB) 2025-12-24 EP disclosed
EP-4667467-A1 PROTAC DEGRADERS OF MLLT1 AND/OR MLLT3 Dark Blue Therapeutics Ltd (GB) 2025-12-24 EP disclosed
WO-2025217121-A1 NOVEL LIPIDS FOR DELIVERY OF NUCLEIC ACID THERAPEUTICS POPVAX PRIVATE LIMITED (IN) 2025-10-16 WO disclosed
US-4281019-A 4-[(Unsaturated or cyclopropylated alkyl)amino]phenyl compounds useful as hypolipidemic and antiatherosclerotic agents AMERICAN CYANAMID COMPANY (US) 1981-07-28 US disclosed
US-4259352-A 4-[Cycloalkyl- or cycloalkenyl-amino(cycloalkyl- or cycloalkenyl-alkenyl)amino]phenyl compounds, useful as hypolipidemic and antiatherosclerotic agents AMERICAN CYANAMID COMPANY (US) 1981-03-31 US disclosed
US-4226878-A ANTIINFLAMMATORY, HYPOTENSIVES, ANTIHISTAMINES KISSEI PHARMACEUTICAL CO., LTD. (JP) 1980-10-07 US disclosed
US-4211783-A Hypolipidemic and antiatherosclerotic novel 4-(aralkyl- and heteroarylalkylamino)phenyl compounds AMERICAN CYANAMID COMPANY (US) 1980-07-08 US disclosed
US-4205085-A Hypolipidemic and antiatherosclerotic 4-(polyfluoroalkylamino)phenyl compounds AMERICAN CYANAMID COMPANY (US) 1980-05-27 US disclosed
EP-0003663-A2 Amino-substituted phenyl and heteroaryl compounds, process for their preparation and pharmaceutical compositions containing them AMERICAN CYANAMID COMPANY (US) 1979-08-22 EP disclosed
US-4107188-A FOR DECREASING LIPID LEVELS HOFFMANN-LA ROCHE INC. (US) 1978-08-15 US disclosed
US-4053618-A ANTILIPOLYTIC ROUSSEL-UCLAF (FR) 1977-10-11 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130261327-A1 METHOD FOR PRODUCING SANSHOOL SCO2, FTH1, CNKSR1 MAPT 4345/4885HCAR2 1059/4885ALDH1A1 1678/4885
US-12570672-B2 Macrocyclic compounds and methods of use KRAS, NRAS, BRAF MAPT 3706/4885HCAR2 4860/4885ALDH1A1 3351/4885
US-20260116838-A1 NEOCARZILIN DERIVATIVES AS ANTIMETASTATIC AGENTS SLC75A1, SLC18A3, SLC8A1 MAPT 1277/4885HCAR2 1249/4885ALDH1A1 756/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.