SCHEMBL6880673

SCHEMBL6880673

CCOC(=O)CCc1ccc(NC(=O)c2cc(-c3ccc(OC(F)(F)F)cc3)cs2)cc1

nearest known ligand 0.58

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MMP12 P39900 5/20 0.58
ABL1 P00519 2/20 0.52
MAPT P10636 2/20 0.47
MMP13 P45452 1/20 0.47
POLB P06746 2/20 0.47
SCN10A Q9Y5Y9 4/20 0.45
ALDH1A1 P00352 1/20 0.43
LMNA P02545 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
FLT1 P17948 1/20 0.42
KDR P35968 1/20 0.42
SYK P43405 1/20 0.42
EPHX2 P34913 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8342310 0.91 MMP12 (0.59) MMP12ABL1MAPTMMP13POLB
SCHEMBL6875530 0.89 MMP12 (0.58) MMP12ABL1MMP13POLBALDH1A1
SCHEMBL6450855 0.88 MMP12 (0.55) MMP12ABL1MMP13SCN10AEPHX2
SCHEMBL6879609 0.87 MMP12 (0.54) MMP12ABL1MAPTMMP13POLB
SCHEMBL6879537 0.83 MMP12 (0.55) MMP12ABL1MAPTMMP13POLB
SCHEMBL6875475 0.83 MMP12 (0.52) MMP12ABL1MAPTMMP13POLB
SCHEMBL8342633 0.83 MMP12 (0.52) MMP12ABL1MAPTMMP13POLB
SCHEMBL6463245 0.81 MMP12 (0.56) MMP12ABL1MMP13SCN10AALDH1A1
SCHEMBL6881932 0.79 MMP12 (0.59) MMP12ABL1MAPTMMP13POLB
SCHEMBL6882916 0.79 MMP12 (0.55) MMP12ABL1MAPTMMP13POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040072871-A1 Novel thiophene derivatives, their process of preparation and the pharmaceutical compositions which comprise them WARNER-LAMBERT COMPANY LLC 2004-04-15 US claimed
US-20040072871-A1 Novel thiophene derivatives, their process of preparation and the pharmaceutical compositions which comprise them WARNER-LAMBERT COMPANY LLC 2004-04-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040072871-A1 Novel thiophene derivatives, their process of preparation and the pharmaceutical compositions which comprise them MMP11, MMP13, CBR1 MMP12 7/4885ABL1 2800/4885MAPT 3516/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.