SCHEMBL6882033

SCHEMBL6882033

O=C(NCc1ccc(F)cc1C(F)(F)F)c1nc(-c2c(F)cccc2F)[nH]c(=O)c1CO

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 10/20 0.42
EPHX2 P34913 6/20 0.39
PPARG P37231 4/20 0.39
HDAC3 O15379 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC2 Q92769 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
NTRK1 P04629 1/20 0.39
ALOX5 P09917 1/20 0.38
ERCC1 P07992 1/20 0.37
FEN1 P39748 1/20 0.37
ERCC4 Q92889 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6885309 0.84 P2RX7 (0.41) P2RX7PPARGERCC1FEN1ERCC4
SCHEMBL6882914 0.82 TACR1 (0.45) ERCC1FEN1ERCC4
SCHEMBL6017784 0.73 P2RX7 (0.45) P2RX7EPHX2PPARGNTRK1ALOX5
SCHEMBL6882031 0.73 SLC6A4 (0.36) ERCC1FEN1ERCC4
SCHEMBL6884591 0.72 ERCC1 (0.50) PPARGERCC1FEN1ERCC4
SCHEMBL15560763 0.70 EPHX2 (0.43) P2RX7EPHX2PPARGNTRK1
SCHEMBL6651068 0.68 ERCC1 (0.52) ERCC1FEN1ERCC4
SCHEMBL18257284 0.67 AR (0.46) P2RX7EPHX2PPARGNTRK1ALOX5
SCHEMBL12641933 0.67 HDAC3 (0.52) P2RX7EPHX2PPARGHDAC3HDAC1
SCHEMBL6355022 0.67 EPHX2 (0.53) P2RX7EPHX2PPARGHDAC3HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004096128-A2 HIV INTEGRASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2004-11-11 WO claimed