SCHEMBL6884591

SCHEMBL6884591

COc1cccc(OC)c1-c1nc(C(=O)NCc2ccc(F)cc2)c(CO)c(=O)[nH]1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERCC1 P07992 1/20 0.50
FEN1 P39748 1/20 0.50
ERCC4 Q92889 1/20 0.50
TDP1 Q9NUW8 1/20 0.46
ALDH1A1 P00352 1/20 0.43
MAPT P10636 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
CNR2 P34972 2/20 0.43
POLB P06746 2/20 0.43
KMT2A Q03164 2/20 0.43
EGLN1 Q9GZT9 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.42
TNKS O95271 1/20 0.42
TNKS2 Q9H2K2 1/20 0.42
PARP2 Q9UGN5 1/20 0.42
APLNR P35414 1/20 0.41
MMP13 P45452 1/20 0.41
ADORA2A P29274 1/20 0.40
MEN1 O00255 1/20 0.40
PPARG P37231 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6017819 0.87 LMNA (0.48) CNR2SMN1; SMN2MMP13ADORA2A
SCHEMBL6651068 0.81 ERCC1 (0.52) ERCC1FEN1ERCC4EGLN1SMN1; SMN2
SCHEMBL6649380 0.78 ERCC1 (0.54) ERCC1FEN1ERCC4EGLN1SMN1; SMN2
SCHEMBL5645281 0.77 ERCC1 (0.42) ERCC1FEN1ERCC4TDP1ALDH1A1
SCHEMBL7156067 0.77 ERCC1 (0.47) ERCC1FEN1ERCC4KMT2AEGLN1
SCHEMBL6885131 0.76 ERCC1 (0.46) ERCC1FEN1ERCC4TDP1ALDH1A1
SCHEMBL6883227 0.76 ERCC1 (0.47) ERCC1FEN1ERCC4ALDH1A1MAPT
SCHEMBL6885309 0.74 P2RX7 (0.41) ERCC1FEN1ERCC4MMP13PPARG
SCHEMBL3534739 0.74 ERCC1 (0.47) ERCC1FEN1ERCC4SMN1; SMN2ADORA2A
SCHEMBL6645591 0.74 ERCC1 (0.47) ERCC1FEN1ERCC4SMN1; SMN2TNKS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004096128-A2 HIV INTEGRASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2004-11-11 WO disclosed