SCHEMBL6885309

SCHEMBL6885309

O=C(NCc1ccc(C(F)(F)F)c(F)c1)c1nc(-c2c(F)cccc2F)[nH]c(=O)c1CO

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 1/20 0.41
PTGER4 P35408 1/20 0.41
ERCC1 P07992 1/20 0.40
FEN1 P39748 1/20 0.40
ERCC4 Q92889 1/20 0.40
HCRTR1 O43613 1/20 0.38
HCRTR2 O43614 1/20 0.38
PTGES O14684 2/20 0.38
PPARG P37231 1/20 0.37
PPARD Q03181 1/20 0.37
PPARA Q07869 1/20 0.37
PDE2A O00408 1/20 0.37
MMP13 P45452 2/20 0.37
CD38 P28907 3/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6882914 0.87 TACR1 (0.45) ERCC1FEN1ERCC4PDE2A
SCHEMBL6882033 0.84 P2RX7 (0.42) P2RX7ERCC1FEN1ERCC4PPARG
SCHEMBL6884591 0.74 ERCC1 (0.50) ERCC1FEN1ERCC4PPARGMMP13
SCHEMBL6018064 0.72 KCNE1 (0.44) P2RX7PTGER4HCRTR1HCRTR2PPARG
SCHEMBL6884192 0.72 PIN1 (0.37) ERCC1FEN1ERCC4
SCHEMBL6017819 0.72 LMNA (0.48) PTGESMMP13
SCHEMBL6651068 0.70 ERCC1 (0.52) ERCC1FEN1ERCC4PDE2A
SCHEMBL4235813 0.67 PTGER4 (0.45) P2RX7PTGER4HCRTR1HCRTR2PTGES
SCHEMBL6649380 0.67 ERCC1 (0.54) ERCC1FEN1ERCC4PDE2A
SCHEMBL6885131 0.67 ERCC1 (0.46) ERCC1FEN1ERCC4PTGES

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004096128-A2 HIV INTEGRASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2004-11-11 WO claimed
WO-2004096128-A2 HIV INTEGRASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2004-11-11 WO disclosed