SCHEMBL6882653

SCHEMBL6882653

CC(NC(=O)c1c[c]ccc1N)c1ccccc1

nearest known ligand 0.69

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.69
KDM4E B2RXH2 4/20 0.69
HPGD P15428 4/20 0.55
LMNA P02545 3/20 0.55
HSD17B10 Q99714 2/20 0.55
POLB P06746 2/20 0.49
L3MBTL1 Q9Y468 1/20 0.49
HDAC3 O15379 1/20 0.49
HDAC4 P56524 1/20 0.49
HDAC1 Q13547 1/20 0.49
HDAC6 Q9UBN7 1/20 0.48
NPC1 O15118 1/20 0.47
CNR1 P21554 1/20 0.46
CNR2 P34972 1/20 0.46
THRB P10828 1/20 0.45
MAPK8 P45983 1/20 0.44
TACR3 P29371 1/20 0.44
KMT2A Q03164 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4278021 0.82 ALDH1A1 (1.00) ALDH1A1KDM4EHPGDLMNAHSD17B10
SCHEMBL4278016 0.82 ALDH1A1 (1.00) ALDH1A1KDM4EHPGDLMNAHSD17B10
SCHEMBL4290720 0.82 ALDH1A1 (1.00) ALDH1A1KDM4EHPGDLMNAHSD17B10
SCHEMBL7023828 0.78 CTSD (0.45) ALDH1A1KDM4EPOLBL3MBTL1HDAC3
SCHEMBL14797294 0.76 ALDH1A1 (0.67) ALDH1A1KDM4EHPGDLMNAHSD17B10
SCHEMBL9953588 0.75 POLB (0.75) ALDH1A1KDM4EHPGDLMNAHSD17B10
SCHEMBL9953590 0.75 POLB (0.75) ALDH1A1KDM4EHPGDLMNAHSD17B10
SCHEMBL9953592 0.75 POLB (0.75) ALDH1A1KDM4EHPGDLMNAHSD17B10
SCHEMBL7431514 0.73 ALDH1A1 (0.62) ALDH1A1KDM4EHPGDLMNAHSD17B10
SCHEMBL7156234 0.73 ALDH1A1 (0.62) ALDH1A1KDM4EHPGDLMNAHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2004505014-A 2004-02-19 JP claimed
EP-1268463-A2 POLYCYCLIC ARYL AND HETEROARYL SUBSTITUTED 4-PYRONES USEFUL FOR SELECTIVE INHIBITION OF THE COAGULATION CASCADE Pharmacia Corporation (US) 2003-01-02 EP claimed
WO-2001077097-A2 POLYCYCLIC ARYL AND HETEROARYL SUBSTITUTED 4-PYRONES USEFUL FOR SELECTIVE INHIBITION OF THE COAGULATION CASCADE PHARMACIA CORPORATION (US) 2001-10-18 WO claimed