SCHEMBL688277

SCHEMBL688277

Cc1ccc([C@H](CC(=O)O)NC(=O)Nc2c(O)ccn(Cc3cccc(S(C)(=O)=O)c3)c2=O)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
POLB P06746 1/20 0.39
HSD17B13 Q7Z5P4 1/20 0.37
CTSA P10619 2/20 0.36
ITGB1 P05556 4/20 0.36
ITGA4 P13612 4/20 0.36
CYP26A1 O43174 2/20 0.36
KEAP1 Q14145 2/20 0.35
NFE2L2 Q16236 2/20 0.35
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
CYP2C9 P11712 1/20 0.35
HPGD P15428 1/20 0.35
CYP2C19 P33261 1/20 0.35
ADRA1D P25100 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.34
LMNA P02545 1/20 0.34
ATM Q13315 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL688357 0.91 POLB (0.41) MEN1KMT2APOLBCTSAITGB1
SCHEMBL688110 0.89 MEN1 (0.49) MEN1KMT2APOLBCTSAITGB1
SCHEMBL687932 0.88 EGLN1 (0.44) MEN1KMT2APOLBCTSAITGB1
SCHEMBL687511 0.87 MEN1 (0.46) MEN1KMT2APOLBCTSAITGB1
SCHEMBL686843 0.87 MAPT (0.47) MEN1KMT2APOLBCTSAKDM4E
SCHEMBL688248 0.87 POLB (0.39) MEN1KMT2APOLBCTSAITGB1
SCHEMBL688150 0.86 ITGB1 (0.38) POLBCTSAITGB1ITGA4CYP26A1
SCHEMBL687488 0.86 MAPT (0.51) MEN1KMT2APOLBCTSAKDM4E
SCHEMBL687925 0.86 CYP26A1 (0.42) MEN1KMT2APOLBCTSAITGB1
SCHEMBL688854 0.84 PPARG (0.39) MEN1KMT2APOLBHSD17B13CTSA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1203766-B1 Carboxylic acid derivatives that inhibit the binding of integrins to their receptors ENCYSIVE PHARMACEUTICALS INC (US) 2012-02-29 EP disclosed
EP-1203766-A2 Carboxylic acid derivatives that inhibit the binding of integrins to their receptors TEXAS BIOTECHNOLOGY CORPORATION (US) 2002-05-08 EP disclosed