SCHEMBL6883124

SCHEMBL6883124

C1=C(Nc2ccnc(-c3ccccc3)n2)OCO1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCG2 Q9UNQ0 1/20 0.48
ITK Q08881 1/20 0.47
MEN1 O00255 7/20 0.43
KMT2A Q03164 7/20 0.43
MAPT P10636 5/20 0.43
KDM4E B2RXH2 4/20 0.43
SMN1; SMN2 Q16637 3/20 0.43
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
POLB P06746 1/20 0.43
CLK4 Q9HAZ1 11/20 0.42
CYP1A2 P05177 11/20 0.42
CYP3A4 P08684 11/20 0.42
CYP2D6 P10635 11/20 0.42
CYP2C19 P33261 10/20 0.42
TP53 P04637 5/20 0.42
TSHR P16473 4/20 0.42
DYRK1A Q13627 3/20 0.42
TDP1 Q9NUW8 2/20 0.42
USP2 O75604 7/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5192222 0.78 LMNA (0.43) ABCG2MEN1KMT2AMAPTNPC1
SCHEMBL3370926 0.77 MEN1 (0.43) MEN1KMT2AMAPTKDM4ESMN1; SMN2
SCHEMBL6883128 0.75 ABCG2 (0.48) ABCG2ITKMEN1KMT2AMAPT
SCHEMBL2422608 0.74 ABCG2 (0.72) ABCG2ITKMEN1KMT2AMAPT
SCHEMBL8346049 0.70 ABCG2 (0.67) ABCG2ITKMEN1KMT2AMAPT
SCHEMBL5261585 0.69 CYP1A2 (0.62) ABCG2ITKMEN1KMT2AMAPT
SCHEMBL11481156 0.68 ADRA2A (0.57) ABCG2ITKMEN1KMT2ASMN1; SMN2
Hydrochloric Acid SCHEMBL5914224 0.67 CYP1A2 (0.60) ABCG2ITKMEN1KMT2AMAPT
SCHEMBL16926442 0.67 ITK (0.57) ABCG2ITKMEN1KMT2ASMN1; SMN2
SCHEMBL21016714 0.66 ITK (0.52) ABCG2ITKMEN1KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003068757-A9 NOVEL PYRIDIN- AND PYRIMIDIN-DERIVATIVES HOFFMANN LA ROCHE (CH) 2004-10-07 WO disclosed