SCHEMBL688327

SCHEMBL688327

Cc1cn(Cc2c(C)cccc2Cl)c(=O)c(NC(=O)N[C@@H](CC(=O)O)c2ccc3c(ccn3C)c2)c1O

nearest known ligand 0.34

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SLC22A12 Q96S37 4/20 0.34
ITGB1 P05556 7/20 0.33
ITGA4 P13612 7/20 0.33
PYGL P06737 1/20 0.33
ITGB7 P26010 1/20 0.33
CTSA P10619 2/20 0.33
CYP26A1 O43174 1/20 0.33
KDM4E B2RXH2 2/20 0.32
ALDH1A1 P00352 2/20 0.32
NOTUM Q6P988 1/20 0.32
HPGD P15428 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL687950 0.91 SMN1; SMN2 (0.36) SLC22A12ITGB1ITGA4CTSAKDM4E
SCHEMBL687687 0.90 PTGER3 (0.38) SLC22A12ITGB1ITGA4CYP26A1NOTUM
SCHEMBL688220 0.88 SLC22A12 (0.36) SLC22A12ITGB1ITGA4PYGLCTSA
SCHEMBL687656 0.86 MEN1 (0.36) ITGB1ITGA4PYGLITGB7CTSA
SCHEMBL688146 0.86 CTSA (0.41) SLC22A12CTSACYP26A1KDM4EALDH1A1
SCHEMBL687310 0.86 CTSA (0.39) PYGLCTSAKDM4EALDH1A1HPGD
SCHEMBL687366 0.85 CTSA (0.37) SLC22A12ITGB1ITGA4CTSAKDM4E
SCHEMBL688079 0.84 PTGER3 (0.38) SLC22A12ITGB1ITGA4CTSACYP26A1
SCHEMBL687082 0.84 POLB (0.39) ITGB1ITGA4CTSACYP26A1KDM4E
SCHEMBL688167 0.83 SMN1; SMN2 (0.43) ITGB1ITGA4CTSAKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1203766-B1 Carboxylic acid derivatives that inhibit the binding of integrins to their receptors ENCYSIVE PHARMACEUTICALS INC (US) 2012-02-29 EP disclosed
EP-1203766-A2 Carboxylic acid derivatives that inhibit the binding of integrins to their receptors TEXAS BIOTECHNOLOGY CORPORATION (US) 2002-05-08 EP disclosed