SCHEMBL687310

SCHEMBL687310

COc1ccc2cc(C(CC(=O)O)NC(=O)Nc3c(O)c(C)cn(Cc4c(C)cccc4Cl)c3=O)ccc2c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSA P10619 6/20 0.39
PTGER3 P43115 3/20 0.38
CYP2C9 P11712 2/20 0.38
CYP2C19 P33261 2/20 0.38
CYP1A2 P05177 1/20 0.38
PDE4A P27815 1/20 0.36
PDE4B Q07343 1/20 0.36
PDE4C Q08493 1/20 0.36
PDE4D Q08499 1/20 0.36
ALDH1A1 P00352 2/20 0.36
KDM4E B2RXH2 1/20 0.36
CYP3A4 P08684 1/20 0.36
GCGR P47871 1/20 0.36
MEN1 O00255 1/20 0.36
MAPT P10636 1/20 0.36
KMT2A Q03164 1/20 0.36
UTS2R Q9UKP6 1/20 0.35
PYGL P06737 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
POLB P06746 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL688330 0.92 SMN1; SMN2 (0.40) CTSAPTGER3CYP2C9CYP2C19CYP1A2
SCHEMBL686938 0.90 PTGER3 (0.47) CTSAPTGER3ALDH1A1GCGRTHRB
SCHEMBL687082 0.89 POLB (0.39) CTSACYP2C9CYP2C19PDE4AALDH1A1
SCHEMBL688220 0.88 SLC22A12 (0.36) CTSACYP2C9CYP2C19ALDH1A1KDM4E
SCHEMBL687907 0.87 SMN1; SMN2 (0.38) CTSAPTGER3ALDH1A1KDM4EMAPT
SCHEMBL688146 0.87 CTSA (0.41) CTSACYP2C9CYP2C19ALDH1A1KDM4E
SCHEMBL693144 0.86 KDM4E (0.37) CTSACYP2C9CYP2C19ALDH1A1KDM4E
SCHEMBL688327 0.86 SLC22A12 (0.34) CTSACYP2C9CYP2C19ALDH1A1KDM4E
SCHEMBL13120941 0.85 ALDH1A1 (0.40) PTGER3CYP2C9CYP2C19CYP1A2ALDH1A1
SCHEMBL688167 0.85 SMN1; SMN2 (0.43) CTSACYP2C9CYP2C19PDE4APDE4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1203766-B1 Carboxylic acid derivatives that inhibit the binding of integrins to their receptors ENCYSIVE PHARMACEUTICALS INC (US) 2012-02-29 EP disclosed
EP-1203766-A2 Carboxylic acid derivatives that inhibit the binding of integrins to their receptors TEXAS BIOTECHNOLOGY CORPORATION (US) 2002-05-08 EP disclosed