SCHEMBL6885488

SCHEMBL6885488

CN(Cc1ccc(F)cc1)C(=O)c1nc(-c2cccnc2)[nH]c(=O)c1O

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PIN1 Q13526 2/20 0.47
ERCC1 P07992 4/20 0.43
FEN1 P39748 4/20 0.43
ERCC4 Q92889 4/20 0.43
GRM1 Q13255 1/20 0.42
RNASEH1 O60930 1/20 0.42
HPGD P15428 1/20 0.40
MAPT P10636 1/20 0.40
KDM4C Q9H3R0 1/20 0.40
CYP11B1 P15538 1/20 0.39
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6885410 0.89 PIN1 (0.60) PIN1ERCC1FEN1ERCC4RNASEH1
SCHEMBL6886274 0.88 ALOX5 (0.49) PIN1ERCC1FEN1ERCC4RNASEH1
SCHEMBL6883330 0.87 PIN1 (0.44) PIN1ERCC1FEN1ERCC4RNASEH1
SCHEMBL6886336 0.86 PIN1 (0.44) PIN1ERCC1FEN1ERCC4RNASEH1
SCHEMBL6649378 0.85 ERCC1 (0.58) PIN1ERCC1FEN1ERCC4RNASEH1
SCHEMBL6883344 0.84 PIN1 (0.43) PIN1ERCC1FEN1ERCC4RNASEH1
SCHEMBL6646945 0.84 ERCC1 (0.50) PIN1ERCC1FEN1ERCC4RNASEH1
SCHEMBL6651065 0.82 ERCC1 (0.51) PIN1ERCC1FEN1ERCC4RNASEH1
SCHEMBL6884647 0.82 ERCC1 (0.43) PIN1ERCC1FEN1ERCC4
SCHEMBL6885301 0.82 PIN1 (0.47) PIN1ERCC1FEN1ERCC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004096128-A2 HIV INTEGRASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2004-11-11 WO claimed
WO-2004096128-A2 HIV INTEGRASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2004-11-11 WO disclosed