SCHEMBL6885301

SCHEMBL6885301

COc1cccc(-c2nc(C(=O)N(C)Cc3ccc(F)cc3)c(O)c(=O)[nH]2)c1

nearest known ligand 0.51

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PIN1 Q13526 3/20 0.47
HSD17B2 P37059 4/20 0.45
ERCC1 P07992 1/20 0.43
FEN1 P39748 1/20 0.43
ERCC4 Q92889 1/20 0.43
HSD17B1 P14061 1/20 0.43
KMT2A Q03164 2/20 0.43
MEN1 O00255 1/20 0.43
ROCK2 O75116 1/20 0.42
ROCK1 Q13464 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6883972 0.88 PIN1 (0.48) PIN1HSD17B2ERCC1FEN1ERCC4
SCHEMBL6877071 0.87 PIN1 (0.47) PIN1HSD17B2ERCC1FEN1ERCC4
SCHEMBL6885410 0.86 PIN1 (0.60) PIN1ERCC1FEN1ERCC4
SCHEMBL6883598 0.85 TNKS (0.43) PIN1ERCC1FEN1ERCC4KMT2A
SCHEMBL6649378 0.82 ERCC1 (0.58) PIN1ERCC1FEN1ERCC4
SCHEMBL6884321 0.82 HSD17B1 (0.44) PIN1HSD17B2ERCC1FEN1ERCC4
SCHEMBL6885488 0.82 PIN1 (0.47) PIN1ERCC1FEN1ERCC4
SCHEMBL6884647 0.81 ERCC1 (0.43) PIN1ERCC1FEN1ERCC4
SCHEMBL6886274 0.81 ALOX5 (0.49) PIN1ERCC1FEN1ERCC4
SCHEMBL6646945 0.81 ERCC1 (0.50) PIN1ERCC1FEN1ERCC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004096128-A2 HIV INTEGRASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2004-11-11 WO claimed
WO-2004096128-A2 HIV INTEGRASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2004-11-11 WO disclosed