SCHEMBL688598

SCHEMBL688598

Cc1ccc([C@H](CC(=O)O)NC(=O)Nc2c(O)ccn(Cc3ccccc3OC(F)F)c2=O)cc1

nearest known ligand 0.39

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.39
CTSA P10619 12/20 0.38
LMNA P02545 2/20 0.37
MAPT P10636 1/20 0.35
PTGER3 P43115 1/20 0.35
MEN1 O00255 1/20 0.34
POLB P06746 1/20 0.34
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL687559 0.91 ALDH1A1 (0.49) ALDH1A1CTSALMNAPTGER3POLB
SCHEMBL687809 0.89 ITGB1 (0.39) ALDH1A1CTSALMNA
SCHEMBL687761 0.87 CTSA (0.46) ALDH1A1CTSALMNAMAPTPTGER3
SCHEMBL687280 0.87 POLB (0.43) CTSALMNAMAPTPTGER3MEN1
SCHEMBL688155 0.85 PTGER3 (0.49) ALDH1A1CTSAMAPTPTGER3MEN1
SCHEMBL688040 0.85 PTGER3 (0.49) ALDH1A1CTSAMAPTPTGER3MEN1
SCHEMBL688191 0.85 ALDH1A1 (0.40) ALDH1A1CTSAPTGER3MEN1POLB
SCHEMBL688132 0.85 TP53 (0.44) ALDH1A1CTSAPTGER3MEN1POLB
SCHEMBL688110 0.84 MEN1 (0.49) ALDH1A1CTSALMNAMAPTMEN1
SCHEMBL688296 0.84 CTSA (0.37) ALDH1A1CTSAPTGER3MEN1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1203766-B1 Carboxylic acid derivatives that inhibit the binding of integrins to their receptors ENCYSIVE PHARMACEUTICALS INC (US) 2012-02-29 EP disclosed
EP-1203766-A2 Carboxylic acid derivatives that inhibit the binding of integrins to their receptors TEXAS BIOTECHNOLOGY CORPORATION (US) 2002-05-08 EP disclosed