SCHEMBL687809

SCHEMBL687809

Cc1ccc([C@H](CC(=O)O)NC(=O)Nc2c(O)ccn(Cc3ccccc3OC(F)(F)F)c2=O)cc1

nearest known ligand 0.39

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 2/20 0.39
ITGA4 P13612 2/20 0.39
ALDH1A1 P00352 1/20 0.39
HSD17B13 Q7Z5P4 6/20 0.39
NTRK1 P04629 2/20 0.38
CTSA P10619 7/20 0.38
LMNA P02545 1/20 0.36
TP53 P04637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL687559 0.90 ALDH1A1 (0.49) ALDH1A1CTSALMNA
SCHEMBL688598 0.89 ALDH1A1 (0.39) ALDH1A1CTSALMNA
SCHEMBL688132 0.88 TP53 (0.44) ALDH1A1NTRK1CTSATP53
SCHEMBL687761 0.87 CTSA (0.46) ALDH1A1CTSALMNATP53
SCHEMBL687280 0.86 POLB (0.43) ITGB1ITGA4CTSALMNA
SCHEMBL688377 0.85 LMNA (0.42) ITGB1ITGA4LMNATP53
SCHEMBL688155 0.85 PTGER3 (0.49) ALDH1A1CTSA
SCHEMBL688040 0.85 PTGER3 (0.49) ALDH1A1CTSA
SCHEMBL688191 0.85 ALDH1A1 (0.40) ITGB1ITGA4ALDH1A1CTSA
SCHEMBL687369 0.84 WDR5 (0.44) ITGB1ITGA4ALDH1A1HSD17B13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1203766-B1 Carboxylic acid derivatives that inhibit the binding of integrins to their receptors ENCYSIVE PHARMACEUTICALS INC (US) 2012-02-29 EP disclosed
EP-1203766-A2 Carboxylic acid derivatives that inhibit the binding of integrins to their receptors TEXAS BIOTECHNOLOGY CORPORATION (US) 2002-05-08 EP disclosed