SCHEMBL6887350

SCHEMBL6887350

CCOC(=O)c1nc(NC(C)=O)sc1Br

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.61
HPGD P15428 1/20 0.61
MEN1 O00255 3/20 0.55
KMT2A Q03164 3/20 0.55
GAA P10253 2/20 0.55
SMN1; SMN2 Q16637 4/20 0.51
NPC1 O15118 3/20 0.51
CYP1A2 P05177 2/20 0.51
RAB9A P51151 2/20 0.51
STAT1 P42224 1/20 0.51
CYP2C9 P11712 1/20 0.51
CYP2C19 P33261 1/20 0.51
TSHR P16473 3/20 0.50
ALOX15 P16050 1/20 0.43
CDK1 P06493 2/20 0.43
CDK4 P11802 2/20 0.43
CCNE1 P24864 2/20 0.43
CDK2 P24941 2/20 0.43
LMNA P02545 3/20 0.42
KDM4E B2RXH2 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1450929 0.84 PIK3CA (0.47) ALDH1A1HPGDMEN1KMT2AGAA
SCHEMBL29019241 0.82 MEN1 (0.50) ALDH1A1HPGDMEN1KMT2AGAA
SCHEMBL4522970 0.82 ALDH1A1 (0.69) ALDH1A1HPGDMEN1KMT2AGAA
SCHEMBL4525950 0.81 ALDH1A1 (0.63) ALDH1A1HPGDMEN1KMT2AGAA
SCHEMBL8726638 0.79 ALDH1A1 (0.51) ALDH1A1HPGDMEN1KMT2AGAA
SCHEMBL6931770 0.78 ALDH1A1 (0.52) ALDH1A1HPGDMEN1KMT2AGAA
SCHEMBL3313992 0.78 ALDH1A1 (0.50) ALDH1A1HPGDMEN1KMT2AGAA
SCHEMBL27760073 0.77 ALDH1A1 (0.51) ALDH1A1HPGDMEN1KMT2AGAA
SCHEMBL12464192 0.77 ALDH1A1 (0.58) ALDH1A1HPGDMEN1KMT2AGAA
SCHEMBL28733816 0.77 ALDH1A1 (0.54) ALDH1A1HPGDMEN1KMT2AGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114450283-B 3, 6-Diamino-pyridazin-3-yl derivatives, pharmaceutical compositions containing them and their use as pro-apoptotic agents 法国施维雅药厂 2024-05-07 CN disclosed
CN-114450284-B 6, 7-Dihydro-5H-pyrido [2,3-C ] pyridazine derivatives as BCL-XL protein inhibitors 法国施维雅药厂 2024-05-07 CN disclosed
CN-114450284-A 6, 7-dihydro-5H-pyrido [2,3-C ] pyridazine derivatives and related compounds as BCL-XL protein inhibitors and pro-apoptotic agents for the treatment of cancer 法国施维雅药厂 2022-05-06 CN disclosed
CN-114450283-A 3, 6-diamino-pyridazin-3-yl derivatives, pharmaceutical compositions containing them and their use as pro-apoptotic agents 法国施维雅药厂 2022-05-06 CN disclosed
US-20040019219-A1 N-alkylated thiazolium salts and process for their preparation LANXESS DEUTSCHLAND GMBH (DE) 2004-01-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040019219-A1 N-alkylated thiazolium salts and process for their preparation AQP4, AQP1, AQP3 ALDH1A1 3073/4885HPGD 3287/4885MEN1 874/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.