SCHEMBL6887435

SCHEMBL6887435

Cn1c(-c2cccc(N)c2)nc2ccc(N3CCN4CCC3CC4)cc2c1=O

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 3/20 0.43
KCNH2 Q12809 6/20 0.41
ADRA1A P35348 5/20 0.41
HRH3 Q9Y5N1 5/20 0.41
PARG Q86W56 1/20 0.38
CHRNA1 P02708 1/20 0.38
CHRNB2 P17787 1/20 0.38
CHRNB4 P30926 1/20 0.38
CHRNA3 P32297 1/20 0.38
CHRNA4 P43681 1/20 0.38
HTR3A P46098 1/20 0.38
IDO1 P14902 1/20 0.37
TDO2 P48775 1/20 0.37
IDO2 Q6ZQW0 1/20 0.37
KMT2A Q03164 1/20 0.36
BRD4 O60885 1/20 0.35
PTGS2 P35354 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6888683 0.91 CHRNA7 (0.46) CHRNA7KCNH2ADRA1AHRH3PARG
SCHEMBL6887461 0.90 CHRNA7 (0.48) CHRNA7KCNH2ADRA1AHRH3PARG
SCHEMBL6888094 0.89 KDM4E (0.44) CHRNA7KCNH2ADRA1AHRH3PARG
SCHEMBL6887469 0.89 CHRNA7 (0.43) CHRNA7KCNH2ADRA1AHRH3PARG
SCHEMBL11905048 0.86 CHRNA7 (0.41) CHRNA7KCNH2ADRA1AHRH3PARG
SCHEMBL1670209 0.86 ADRA1A (0.42) CHRNA7KCNH2ADRA1AHRH3PARG
SCHEMBL6886312 0.86 HPGD (0.40) CHRNA7BRD4
SCHEMBL6887372 0.84 CHRNA7 (0.47) CHRNA7KCNH2ADRA1AHRH3PARG
SCHEMBL6889957 0.84 HRH3 (0.45) CHRNA7KCNH2ADRA1AHRH3CHRNA1
SCHEMBL6889695 0.83 CHRNA7 (0.38) CHRNA7KCNH2CHRNA1CHRNB2CHRNB4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011045258-A1 CONDENSED AZINE - DERIVATIVES FOR THE TREATMENT OF DISEASES RELATED TO THE ACETYLCHOLINE RECEPTOR N.V. ORGANON (NL) 2011-04-21 WO disclosed