SCHEMBL6888048

SCHEMBL6888048

CCOC(=O)c1ccc(-c2cccc(O)c2)nc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B1 P14061 3/20 0.53
HSD17B2 P37059 3/20 0.53
CSNK1D P48730 1/20 0.50
NPC1 O15118 1/20 0.50
RAB9A P51151 1/20 0.50
JAK2 O60674 1/20 0.50
JAK3 P52333 1/20 0.50
CA12 O43570 3/20 0.49
CA1 P00915 3/20 0.49
CA2 P00918 3/20 0.49
CA7 P43166 3/20 0.49
CA9 Q16790 3/20 0.49
CA14 Q9ULX7 3/20 0.49
ESR1 P03372 1/20 0.49
ESR2 Q92731 1/20 0.49
TP53 P04637 1/20 0.48
MAPT P10636 1/20 0.48
HPGDS O60760 1/20 0.45
CHEK1 O14757 1/20 0.44
FYN P06241 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29596804 0.86 NPC1 (0.52) NPC1RAB9ATP53MAPT
SCHEMBL2009526 0.86 HPGDS (0.64) CSNK1DNPC1RAB9AJAK2JAK3
SCHEMBL851716 0.85 NPC1 (0.51) NPC1RAB9ACA12CA1CA2
SCHEMBL29914699 0.85 HSD17B1 (0.56) HSD17B1HSD17B2CA12CA1CA2
SCHEMBL21228142 0.85 HSD17B1 (0.56) HSD17B1HSD17B2CA12CA1CA2
SCHEMBL1222552 0.85 NPC1 (0.62) NPC1RAB9ATP53MAPTHPGDS
SCHEMBL1749701 0.84 TP53 (0.48) NPC1RAB9ATP53MAPTHPGDS
SCHEMBL2218765 0.82 NPC1 (0.46) NPC1RAB9ATP53MAPTHPGDS
SCHEMBL1749621 0.82 NPC1 (0.46) NPC1RAB9ATP53MAPTHPGDS
SCHEMBL3900684 0.82 NPC1 (0.56) NPC1RAB9ACA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6831106-B1 Selective activity on cell proliferation and differentiation without displaying any hypercalcaemiant nature GALDERMA RESEARCH & DEVELOPMENT, S.N.C. (FR) 2004-12-14 US disclosed