SCHEMBL6888946

SCHEMBL6888946

COC(=O)c1ccc(-c2cccc(O)c2C)cc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 1/20 0.57
CA1 P00915 6/20 0.50
CA2 P00918 6/20 0.50
CA12 O43570 5/20 0.50
CA9 Q16790 5/20 0.50
CA14 Q9ULX7 5/20 0.50
CA7 P43166 3/20 0.50
TDP1 Q9NUW8 1/20 0.50
KDM4A O75164 1/20 0.48
PTPN1 P18031 2/20 0.48
PTPRC P08575 1/20 0.48
PTPRF P10586 1/20 0.48
CDC25B P30305 1/20 0.48
TSHR P16473 1/20 0.47
ERN1 O75460 2/20 0.47
MAPT P10636 3/20 0.46
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
POLB P06746 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29141105 0.85 EGFR (0.59) EGFRCA1CA2CA12CA9
SCHEMBL2035147 0.85 EGFR (0.71) EGFRCA1CA2CA12CA9
SCHEMBL2038076 0.83 EGFR (0.49) EGFRCA1CA2CA12CA9
SCHEMBL29788171 0.83 EGFR (0.49) EGFRCA1CA2CA12CA9
SCHEMBL6566323 0.81 RXRA (0.46) EGFRCA1CA2CA12CA9
SCHEMBL6882126 0.80 CA12 (0.50) EGFRCA1CA2CA12CA9
SCHEMBL6887241 0.78 PDK2 (0.49) EGFRCA1CA2CA12CA9
SCHEMBL3312749 0.78 EGFR (0.58) EGFRCA1CA2CA12CA9
SCHEMBL27708108 0.78 EGFR (0.71) EGFRCA1CA2CA12CA9
SCHEMBL2037520 0.77 NR3C1 (0.57) EGFRCA1CA2CA12CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6831106-B1 Selective activity on cell proliferation and differentiation without displaying any hypercalcaemiant nature GALDERMA RESEARCH & DEVELOPMENT, S.N.C. (FR) 2004-12-14 US disclosed