SCHEMBL6892362

SCHEMBL6892362

Cc1ccc(C(N)=S)c(Br)c1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.39
HPGD P15428 2/20 0.39
RAD52 P43351 1/20 0.39
HTT P42858 3/20 0.38
GAA P10253 2/20 0.38
KDM4E B2RXH2 1/20 0.38
CYP1A2 P05177 2/20 0.36
NPC1 O15118 4/20 0.36
RAB9A P51151 3/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
L3MBTL1 Q9Y468 2/20 0.36
HSP90AA1 P07900 1/20 0.36
MAPT P10636 3/20 0.35
MAPK1 P28482 1/20 0.35
ALOX15 P16050 2/20 0.34
HSD17B10 Q99714 1/20 0.34
CTSL P07711 3/20 0.34
HTR2A P28223 1/20 0.34
HTR2C P28335 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL305165 0.79 ERN1 (0.46) ALDH1A1HPGDHTTGAANPC1
SCHEMBL10147428 0.78 TDP1 (0.44) ALDH1A1HPGDRAD52HTTGAA
SCHEMBL27973657 0.77 ALDH1A1 (0.42) ALDH1A1HPGDRAD52GAAKDM4E
SCHEMBL7168641 0.77 ALDH1A1 (0.50) ALDH1A1HPGDRAD52HTTGAA
SCHEMBL20241764 0.76 ALDH1A1 (0.68) ALDH1A1HPGDRAD52GAAKDM4E
SCHEMBL19096781 0.75 FLT1 (0.42) ALDH1A1HPGDRAD52GAAKDM4E
SCHEMBL6843558 0.75 ALDH1A1 (0.39) ALDH1A1HPGDRAD52HTTGAA
SCHEMBL6897299 0.75 RAB9A (0.47) ALDH1A1HPGDRAD52HTTGAA
SCHEMBL4302622 0.75 ALDH1A1 (0.42) ALDH1A1HPGDRAD52GAANPC1
SCHEMBL14800110 0.74 ALDH1A1 (0.48) ALDH1A1HPGDHTTGAAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1126833-A4 OXADIAZOLE, THIADIAZOLE AND TRIAZOLE DERIVATIVES AND COMBINATORIAL LIBRARIES THEREOF TREGA BIOSCIENCES INC (US) 2004-09-08 EP claimed
EP-1126833-A2 OXADIAZOLE, THIADIAZOLE AND TRIAZOLE DERIVATIVES AND COMBINATORIAL LIBRARIES THEREOF TREGA BIOSCIENCES, INC. (US) 2001-08-29 EP claimed
WO-2000025768-A1 OXADIAZOLE, THIADIAZOLE AND TRIAZOLE DERIVATIVES AND COMBINATORIAL LIBRARIES THEREOF TREGA BIOSCIENCES, INC. (US) 2000-05-11 WO claimed